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Synthesis and biological evaluation of copper-64 radiolabeled [DUPA-6-Ahx-(NODAGA)-5-Ava-BBN(7-14)NH2], a novel bivalent targeting vector having affinity for two distinct biomarkers (GRPr/PSMA) of prostate cancer.
Bandari, Rajendra Prasad; Jiang, Zongrun; Reynolds, Tamila Stott; Bernskoetter, Nicole E; Szczodroski, Ashley F; Bassuner, Kurt J; Kirkpatrick, Daniel L; Rold, Tammy L; Sieckman, Gary L; Hoffman, Timothy J; Connors, James P; Smith, Charles J.
Afiliação
  • Bandari RP; Research Service, Truman VA, Columbia, MO 65201, USA; Department of Radiology, University of Missouri School of Medicine, Columbia, MO 65211, USA.
  • Jiang Z; Research Service, Truman VA, Columbia, MO 65201, USA; Department of Chemistry, University of Missouri, Columbia, MO 65211, USA.
  • Reynolds TS; Research Service, Truman VA, Columbia, MO 65201, USA; Department of Veterinary Pathobiology, University of Missouri College of Veterinary Medicine, Columbia, MO 65211, USA.
  • Bernskoetter NE; Research Service, Truman VA, Columbia, MO 65201, USA; Department of Radiology, University of Missouri School of Medicine, Columbia, MO 65211, USA.
  • Szczodroski AF; Research Service, Truman VA, Columbia, MO 65201, USA.
  • Bassuner KJ; Department of Radiology, University of Missouri School of Medicine, Columbia, MO 65211, USA.
  • Kirkpatrick DL; Department of Radiology, University of Missouri School of Medicine, Columbia, MO 65211, USA.
  • Rold TL; Research Service, Truman VA, Columbia, MO 65201, USA; Department of Internal Medicine, University of Missouri School of Medicine, Columbia, MO 65211, USA.
  • Sieckman GL; Research Service, Truman VA, Columbia, MO 65201, USA.
  • Hoffman TJ; Research Service, Truman VA, Columbia, MO 65201, USA; Department of Internal Medicine, University of Missouri School of Medicine, Columbia, MO 65211, USA; Department of Chemistry, University of Missouri, Columbia, MO 65211, USA.
  • Connors JP; Department of Radiology, University of Missouri School of Medicine, Columbia, MO 65211, USA.
  • Smith CJ; Research Service, Truman VA, Columbia, MO 65201, USA; Department of Radiology, University of Missouri School of Medicine, Columbia, MO 65211, USA; University of Missouri Research Reactor Center, University of Missouri, Columbia, MO 65211, USA. Electronic address: smithcj@health.missouri.edu.
Nucl Med Biol ; 41(4): 355-63, 2014 Apr.
Article em En | MEDLINE | ID: mdl-24508213

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Bombesina / Radioisótopos de Cobre / Biomarcadores Tumorais / Receptores da Bombesina / Glutamato Carboxipeptidase II / Antígenos de Superfície Tipo de estudo: Guideline Limite: Animals / Female / Humans / Male Idioma: En Revista: Nucl Med Biol Assunto da revista: BIOLOGIA / MEDICINA NUCLEAR Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Bombesina / Radioisótopos de Cobre / Biomarcadores Tumorais / Receptores da Bombesina / Glutamato Carboxipeptidase II / Antígenos de Superfície Tipo de estudo: Guideline Limite: Animals / Female / Humans / Male Idioma: En Revista: Nucl Med Biol Assunto da revista: BIOLOGIA / MEDICINA NUCLEAR Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Estados Unidos