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Temozolomide analogs with improved brain/plasma ratios - Exploring the possibility of enhancing the therapeutic index of temozolomide.
Rai, Roopa; Banerjee, Monali; Wong, Darren H; McCullagh, Emma; Gupta, Ashu; Tripathi, Shailendra; Riquelme, Eduardo; Jangir, Ramnivas; Yadav, Shyamraj; Raja, Mohd; Melkani, Pankaj; Dixit, Vikas; Patil, Umesh; Shrivastava, Ritesh; Middya, Sandip; Olivares, Felipe; Guerrero, Javier; Surya, Arjun; Pham, Son M; Bernales, Sebastián; Protter, Andrew A; Hung, David T; Chakravarty, Sarvajit.
Afiliação
  • Rai R; Medivation, 525 Market Street, 36th Floor, San Francisco, CA 94105, USA.
  • Banerjee M; Curadev Pvt. Ltd, B-87, Sector 83, Noida, Uttar Pradesh 201305, India.
  • Wong DH; Concert Pharmaceuticals, 99 Hayden Ave, Suite 500, Lexington, MA 02421, USA.
  • McCullagh E; Medivation, 525 Market Street, 36th Floor, San Francisco, CA 94105, USA.
  • Gupta A; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Tripathi S; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Riquelme E; Fundación Ciencia y Vida, Avenida Zañartu 1482, Ñuñoa, Santiago 7780272, Chile.
  • Jangir R; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Yadav S; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Raja M; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Melkani P; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Dixit V; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Patil U; Integral BioScience Pvt. Ltd, C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Shrivastava R; Curadev Pvt. Ltd, B-87, Sector 83, Noida, Uttar Pradesh 201305, India.
  • Middya S; Curadev Pvt. Ltd, B-87, Sector 83, Noida, Uttar Pradesh 201305, India.
  • Olivares F; Fundación Ciencia y Vida, Avenida Zañartu 1482, Ñuñoa, Santiago 7780272, Chile.
  • Guerrero J; Fundación Ciencia y Vida, Avenida Zañartu 1482, Ñuñoa, Santiago 7780272, Chile.
  • Surya A; Curadev Pvt. Ltd, B-87, Sector 83, Noida, Uttar Pradesh 201305, India.
  • Pham SM; Medivation, 525 Market Street, 36th Floor, San Francisco, CA 94105, USA.
  • Bernales S; Medivation, 525 Market Street, 36th Floor, San Francisco, CA 94105, USA.
  • Protter AA; Medivation, 525 Market Street, 36th Floor, San Francisco, CA 94105, USA.
  • Hung DT; Medivation, 525 Market Street, 36th Floor, San Francisco, CA 94105, USA.
  • Chakravarty S; Medivation, 525 Market Street, 36th Floor, San Francisco, CA 94105, USA.
Bioorg Med Chem Lett ; 26(20): 5103-5109, 2016 10 15.
Article em En | MEDLINE | ID: mdl-27614414

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Encéfalo / Antineoplásicos Alquilantes / Dacarbazina Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Encéfalo / Antineoplásicos Alquilantes / Dacarbazina Tipo de estudo: Prognostic_studies Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2016 Tipo de documento: Article País de afiliação: Estados Unidos