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Structure-guided design, synthesis and evaluation of oxazolidinone-based inhibitors of norovirus 3CL protease.
Damalanka, Vishnu C; Kim, Yunjeong; Galasiti Kankanamalage, Anushka C; Rathnayake, Athri D; Mehzabeen, Nurjahan; Battaile, Kevin P; Lovell, Scott; Nguyen, Harry Nhat; Lushington, Gerald H; Chang, Kyeong-Ok; Groutas, William C.
Afiliação
  • Damalanka VC; Department of Chemistry, Wichita State University, Wichita, KS 67260, USA.
  • Kim Y; Department of Diagnostic Medicine & Pathobiology, College of Veterinary Medicine, Kansas State University, Manhattan, KS 66506, USA.
  • Galasiti Kankanamalage AC; Department of Chemistry, Wichita State University, Wichita, KS 67260, USA.
  • Rathnayake AD; Department of Chemistry, Wichita State University, Wichita, KS 67260, USA.
  • Mehzabeen N; Protein Structure Laboratory, The University of Kansas, Lawrence, KS 66047, USA.
  • Battaile KP; IMCA-CAT, Hauptman-Woodward Medical Research Institute, APS Argonne National Laboratory, Argonne, IL 60439, USA.
  • Lovell S; Protein Structure Laboratory, The University of Kansas, Lawrence, KS 66047, USA.
  • Nguyen HN; Department of Chemistry, Wichita State University, Wichita, KS 67260, USA.
  • Lushington GH; LiS Consulting, Lawrence, KS 66046, USA.
  • Chang KO; Department of Diagnostic Medicine & Pathobiology, College of Veterinary Medicine, Kansas State University, Manhattan, KS 66506, USA. Electronic address: kchang@vet.ksu.edu.
  • Groutas WC; Department of Chemistry, Wichita State University, Wichita, KS 67260, USA. Electronic address: bill.groutas@wichita.edu.
Eur J Med Chem ; 143: 881-890, 2018 Jan 01.
Article em En | MEDLINE | ID: mdl-29227928

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Proteínas Virais / Oxazolidinonas / Norovirus Idioma: En Revista: Eur J Med Chem Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Inibidores de Proteases / Proteínas Virais / Oxazolidinonas / Norovirus Idioma: En Revista: Eur J Med Chem Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos