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Design, synthesis and evaluation of potent and selective inhibitors of mono-(ADP-ribosyl)transferases PARP10 and PARP14.
Holechek, Jacob; Lease, Robert; Thorsell, Ann-Gerd; Karlberg, Tobias; McCadden, Caitlin; Grant, Ryan; Keen, Abby; Callahan, Evan; Schüler, Herwig; Ferraris, Dana.
Afiliação
  • Holechek J; McDaniel College, 2 College Hill, Westminster, MD 21157, United States.
  • Lease R; McDaniel College, 2 College Hill, Westminster, MD 21157, United States.
  • Thorsell AG; Karolinska Institutet, Department of Biosciences and Nutrition, Hälsovägen 7c, S-14157 Huddinge, Sweden.
  • Karlberg T; Karolinska Institutet, Department of Biosciences and Nutrition, Hälsovägen 7c, S-14157 Huddinge, Sweden.
  • McCadden C; McDaniel College, 2 College Hill, Westminster, MD 21157, United States.
  • Grant R; McDaniel College, 2 College Hill, Westminster, MD 21157, United States.
  • Keen A; McDaniel College, 2 College Hill, Westminster, MD 21157, United States.
  • Callahan E; McDaniel College, 2 College Hill, Westminster, MD 21157, United States.
  • Schüler H; Karolinska Institutet, Department of Biosciences and Nutrition, Hälsovägen 7c, S-14157 Huddinge, Sweden.
  • Ferraris D; McDaniel College, 2 College Hill, Westminster, MD 21157, United States. Electronic address: dferraris@mcdaniel.edu.
Bioorg Med Chem Lett ; 28(11): 2050-2054, 2018 06 15.
Article em En | MEDLINE | ID: mdl-29748053

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Proteínas Proto-Oncogênicas / Poli(ADP-Ribose) Polimerases / Éteres / Inibidores de Poli(ADP-Ribose) Polimerases / Amidas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Desenho de Fármacos / Proteínas Proto-Oncogênicas / Poli(ADP-Ribose) Polimerases / Éteres / Inibidores de Poli(ADP-Ribose) Polimerases / Amidas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Estados Unidos