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Virtual screening-driven discovery of dual 5-HT6/5-HT2A receptor ligands with pro-cognitive properties.
Staron, Jakub; Kurczab, Rafal; Warszycki, Dawid; Satala, Grzegorz; Krawczyk, Martyna; Bugno, Ryszard; Lenda, Tomasz; Popik, Piotr; Hogendorf, Adam S; Hogendorf, Agata; Dubiel, Krzysztof; Matloka, Mikolaj; Moszczynski-Petkowski, Rafal; Pieczykolan, Jerzy; Wieczorek, Maciej; Zajdel, Pawel; Bojarski, Andrzej J.
Afiliação
  • Staron J; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland. Electronic address: staron@if-pan.krakow.pl.
  • Kurczab R; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Warszycki D; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Satala G; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Krawczyk M; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Bugno R; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Lenda T; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Popik P; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Hogendorf AS; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Hogendorf A; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
  • Dubiel K; Celon Pharma S.A., 2A Ogrodowa Street, 05-092, Lomianki, Poland.
  • Matloka M; Celon Pharma S.A., 2A Ogrodowa Street, 05-092, Lomianki, Poland.
  • Moszczynski-Petkowski R; Celon Pharma S.A., 2A Ogrodowa Street, 05-092, Lomianki, Poland.
  • Pieczykolan J; Celon Pharma S.A., 2A Ogrodowa Street, 05-092, Lomianki, Poland.
  • Wieczorek M; Celon Pharma S.A., 2A Ogrodowa Street, 05-092, Lomianki, Poland.
  • Zajdel P; Department of Medicinal Chemistry, Jagiellonian University Medical College, 9 Medyczna Street, 30-688, Kraków, Poland.
  • Bojarski AJ; Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343, Kraków, 12 Smetna Street, Poland.
Eur J Med Chem ; 185: 111857, 2020 Jan 01.
Article em En | MEDLINE | ID: mdl-31734022

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antipsicóticos / Triptaminas / Receptores de Serotonina / Cognição / Receptor 5-HT2A de Serotonina / Antidepressivos Tipo de estudo: Diagnostic_studies / Prognostic_studies / Screening_studies Limite: Animals / Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Antipsicóticos / Triptaminas / Receptores de Serotonina / Cognição / Receptor 5-HT2A de Serotonina / Antidepressivos Tipo de estudo: Diagnostic_studies / Prognostic_studies / Screening_studies Limite: Animals / Humans Idioma: En Revista: Eur J Med Chem Ano de publicação: 2020 Tipo de documento: Article