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Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody-Drug Conjugates.
Nicolaou, K C; Li, Ruofan; Chen, Qifeng; Lu, Zhaoyong; Pitsinos, Emmanuel N; Schammel, Alexander; Lin, Baiwei; Gu, Christine; Sarvaiya, Hetal; Tchelepi, Robert; Valdiosera, Amanda; Clubb, Justin; Barbour, Nicole; Sisodiya, Vikram; Sandoval, Joseph; Lee, Christina; Aujay, Monette; Gavrilyuk, Julia.
Afiliação
  • Nicolaou KC; Department of Chemistry, BioScience Research Collaborative, Rice University, 6100 Main Street, Houston, Texas 77005, United States.
  • Li R; Department of Chemistry, BioScience Research Collaborative, Rice University, 6100 Main Street, Houston, Texas 77005, United States.
  • Chen Q; Department of Chemistry, BioScience Research Collaborative, Rice University, 6100 Main Street, Houston, Texas 77005, United States.
  • Lu Z; Department of Chemistry, BioScience Research Collaborative, Rice University, 6100 Main Street, Houston, Texas 77005, United States.
  • Pitsinos EN; Department of Chemistry, BioScience Research Collaborative, Rice University, 6100 Main Street, Houston, Texas 77005, United States.
  • Schammel A; Laboratory of Natural Products Synthesis & Bioorganic Chemistry, Institute of Nanoscience and Nanotechnology, National Centre for Scientific Research "Demokritos", 153 10 Agia Paraskevi, Greece.
  • Lin B; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Gu C; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Sarvaiya H; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Tchelepi R; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Valdiosera A; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Clubb J; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Barbour N; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Sisodiya V; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Sandoval J; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Lee C; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Aujay M; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
  • Gavrilyuk J; AbbVie, Inc., 400 East Jamie Court, South San Francisco, California 94080, United States.
J Am Chem Soc ; 142(29): 12890-12899, 2020 07 22.
Article em En | MEDLINE | ID: mdl-32662641

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Carbolinas / Imunoconjugados / Dissacarídeos / Enedi-Inos / Antineoplásicos Limite: Humans Idioma: En Revista: J Am Chem Soc Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Carbolinas / Imunoconjugados / Dissacarídeos / Enedi-Inos / Antineoplásicos Limite: Humans Idioma: En Revista: J Am Chem Soc Ano de publicação: 2020 Tipo de documento: Article País de afiliação: Estados Unidos