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Positive allosteric mechanisms of adenosine A1 receptor-mediated analgesia.
Draper-Joyce, Christopher J; Bhola, Rebecca; Wang, Jinan; Bhattarai, Apurba; Nguyen, Anh T N; Cowie-Kent, India; O'Sullivan, Kelly; Chia, Ling Yeong; Venugopal, Hariprasad; Valant, Celine; Thal, David M; Wootten, Denise; Panel, Nicolas; Carlsson, Jens; Christie, Macdonald J; White, Paul J; Scammells, Peter; May, Lauren T; Sexton, Patrick M; Danev, Radostin; Miao, Yinglong; Glukhova, Alisa; Imlach, Wendy L; Christopoulos, Arthur.
Afiliação
  • Draper-Joyce CJ; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Bhola R; The Florey Institute of Neuroscience and Mental Health, University of Melbourne, Parkville, Victoria, Australia.
  • Wang J; Department of Physiology, Monash Biomedicine Discovery Institute, Monash University, Clayton, Victoria, Australia.
  • Bhattarai A; Center for Computational Biology and Department of Molecular Biosciences, University of Kansas, Lawrence, KS, USA.
  • Nguyen ATN; Center for Computational Biology and Department of Molecular Biosciences, University of Kansas, Lawrence, KS, USA.
  • Cowie-Kent I; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • O'Sullivan K; Department of Physiology, Monash Biomedicine Discovery Institute, Monash University, Clayton, Victoria, Australia.
  • Chia LY; Department of Physiology, Monash Biomedicine Discovery Institute, Monash University, Clayton, Victoria, Australia.
  • Venugopal H; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Valant C; Department of Biochemistry and Molecular Biology, Monash University, Clayton, Victoria, Australia.
  • Thal DM; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Wootten D; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Panel N; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Carlsson J; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Christie MJ; Science for Life Laboratory, Department of Cell and Molecular Biology, Uppsala University, Uppsala, Sweden.
  • White PJ; Science for Life Laboratory, Department of Cell and Molecular Biology, Uppsala University, Uppsala, Sweden.
  • Scammells P; Discipline of Pharmacology, Faculty of Medicine and Health, University of Sydney, Camperdown, New South Wales, Australia.
  • May LT; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Sexton PM; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Danev R; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Miao Y; Drug Discovery Biology and Department of Pharmacology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Glukhova A; ARC Centre for Cryo-electron Microscopy of Membrane Proteins, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, Victoria, Australia.
  • Imlach WL; Graduate School of Medicine, University of Tokyo, Tokyo, Japan.
  • Christopoulos A; Center for Computational Biology and Department of Molecular Biosciences, University of Kansas, Lawrence, KS, USA.
Nature ; 597(7877): 571-576, 2021 09.
Article em En | MEDLINE | ID: mdl-34497422

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptor A1 de Adenosina / Analgesia Limite: Animals Idioma: En Revista: Nature Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Austrália

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Receptor A1 de Adenosina / Analgesia Limite: Animals Idioma: En Revista: Nature Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Austrália