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Discovery of the c-Jun N-Terminal Kinase Inhibitor CC-90001.
Nagy, Mark A; Hilgraf, Robert; Mortensen, Deborah S; Elsner, Jan; Norris, Stephen; Tikhe, Jayashree; Yoon, Won; Paisner, David; Delgado, Mercedes; Erdman, Paul; Haelewyn, Jason; Khambatta, Godrej; Xu, Li; Romanow, William J; Condroski, Kevin; Bahmanyar, Sogole; McCarrick, Meg; Benish, Brent; Blease, Kate; LeBrun, Laurie; Moghaddam, Mehran F; Apuy, Julius; Canan, Stacie S; Bennett, Brydon L; Satoh, Yoshitaka.
Afiliação
  • Nagy MA; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Hilgraf R; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Mortensen DS; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Elsner J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Norris S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Tikhe J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Yoon W; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Paisner D; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Delgado M; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Erdman P; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Haelewyn J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Khambatta G; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Xu L; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Romanow WJ; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Condroski K; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Bahmanyar S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • McCarrick M; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Benish B; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Blease K; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • LeBrun L; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Moghaddam MF; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Apuy J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Canan SS; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Bennett BL; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Satoh Y; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
J Med Chem ; 64(24): 18193-18208, 2021 12 23.
Article em En | MEDLINE | ID: mdl-34894681

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinas / Cicloexilaminas / Proteínas Quinases JNK Ativadas por Mitógeno / Inibidores de Proteínas Quinases / Descoberta de Drogas Limite: Animals / Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Pirimidinas / Cicloexilaminas / Proteínas Quinases JNK Ativadas por Mitógeno / Inibidores de Proteínas Quinases / Descoberta de Drogas Limite: Animals / Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Estados Unidos