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Identification and in vitro characterization of a new series of potent and highly selective G9a inhibitors as novel anti-fibroadipogenic agents.
Randazzo, Pietro; Sinisi, Roberta; Gornati, Davide; Bertuolo, Stefania; Bencheva, Leda; De Matteo, Marilenia; Nibbio, Martina; Monteagudo, Edith; Turcano, Lorenzo; Bianconi, Valeria; Peruzzi, Giovanna; Summa, Vincenzo; Bresciani, Alberto; Mozzetta, Chiara; Di Fabio, Romano.
Afiliação
  • Randazzo P; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Sinisi R; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Gornati D; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Bertuolo S; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Bencheva L; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • De Matteo M; Promidis, Via Olgettina 60, 20132 Milano, Italy.
  • Nibbio M; IRBM Science Park, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Monteagudo E; CHDI Foundation, 6080 Center Drive, Suite 700, CA 90045, Los Angeles.
  • Turcano L; IRBM Science Park, Via Pontina Km 30.600, 00070 Pomezia, Italy.
  • Bianconi V; Institute of Molecular Biology and Pathology (IBPM), National Research Council (CNR) of Italy c/o, Department of Biology and Biotechnology "C. Darwin", Sapienza University, Piazzale A. Moro 5, 00185 Rome, Italy.
  • Peruzzi G; Center for Life Nano- & Neuro-Science, Fondazione Istituto Italiano di Tecnologia (IIT), V.le Regina, Elena 291, 00161 Rome, Italy.
  • Summa V; University of Naples Federico II, Vial Domenico Montesano 49, 80131, Naples, Italy.
  • Bresciani A; Exscientia LTD, The Schrödinger Building Oxford Science Park, Oxford OX4 4GE, UK.
  • Mozzetta C; Institute of Molecular Biology and Pathology (IBPM), National Research Council (CNR) of Italy c/o, Department of Biology and Biotechnology "C. Darwin", Sapienza University, Piazzale A. Moro 5, 00185 Rome, Italy.
  • Di Fabio R; Promidis, Via Olgettina 60, 20132 Milano, Italy; IRBM Science Park, Via Pontina Km 30.600, 00070 Pomezia, Italy. Electronic address: r.difabio@irbm.com.
Bioorg Med Chem Lett ; 72: 128858, 2022 09 15.
Article em En | MEDLINE | ID: mdl-35718104

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Histonas / Histona-Lisina N-Metiltransferase Tipo de estudo: Diagnostic_studies Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Itália

Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Histonas / Histona-Lisina N-Metiltransferase Tipo de estudo: Diagnostic_studies Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Itália