Atropodiastereoselective 5N-Acylation of 1,5-Benzodiazepin-2-ones with (S)-2-Phenylpropanoyl and (S)-2-Phenylbutanoyl Chlorides.

Funaki, Kaoru; Tabata, Hidetsugu; Nakazato, Yusuke; Takahashi, Yuka; Tasaka, Tomohiko; Takahashi, Hideyo; Natsugari, Hideaki; Oshitari, Tetsuta

Funaki, Kaoru; Tabata, Hidetsugu; Nakazato, Yusuke; Takahashi, Yuka; Tasaka, Tomohiko; Takahashi, Hideyo; Natsugari, Hideaki; Oshitari, Tetsuta.

Afiliação

Funaki K; Faculty of Pharma Sciences, Teikyo University, 2-11-1 Kaga, Itabashi-ku, Tokyo 173-8605, Japan.
Tabata H; Faculty of Pharma Sciences, Teikyo University, 2-11-1 Kaga, Itabashi-ku, Tokyo 173-8605, Japan.
Nakazato Y; Faculty of Pharma Sciences, Teikyo University, 2-11-1 Kaga, Itabashi-ku, Tokyo 173-8605, Japan.
Takahashi Y; Faculty of Pharma Sciences, Teikyo University, 2-11-1 Kaga, Itabashi-ku, Tokyo 173-8605, Japan.
Tasaka T; Affinity Science Corporation, 1-11-1 Nishi-Gotanda, Shinagawa-ku, Tokyo 141-0031, Japan.
Takahashi H; Faculty of Pharmaceutical Sciences, Tokyo University of Science, 2641 Yamazaki, Noda, Chiba 278-8510, Japan.
Natsugari H; Affinity Science Corporation, 1-11-1 Nishi-Gotanda, Shinagawa-ku, Tokyo 141-0031, Japan.
Oshitari T; Faculty of Pharmaceutical Sciences, The University of Tokyo, 7-3-1 Hongo, Bunkyo-ku, Tokyo 113-0033, Japan.

J Org Chem ; 87(22): 15289-15300, 2022 11 18.

Article em En | MEDLINE | ID: mdl-36222058

Assuntos

Benzodiazepinas; Cloretos; Benzeno/química; Acilação

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Texto completo: 1 Coleções: 01-internacional Base de dados: MEDLINE Assunto principal: Benzodiazepinas / Cloretos Idioma: En Revista: J Org Chem Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Japão

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