Detalles de la búsqueda
1.
Novel multifunctional tacrine-donepezil hybrids against Alzheimer's disease: Design synthesis and bioactivity studies.
Arch Pharm (Weinheim);
: e2300575, 2024 Apr 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-38593283
2.
N-Substituted piperidine-3-carbohydrazide-hydrazones against Alzheimer's disease: Synthesis and evaluation of cholinesterase, beta-amyloid inhibitory activity, and antioxidant capacity.
Arch Pharm (Weinheim);
356(3): e2200519, 2023 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-36461719
3.
Design, synthesis, acetylcholinesterase, butyrylcholinesterase, and amyloid-ß aggregation inhibition studies of substituted 4,4'-diimine/4,4'-diazobiphenyl derivatives.
Arch Pharm (Weinheim);
355(12): e2200152, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35976708
4.
Design, synthesis, and in vitro biological evaluation of novel thiazolopyrimidine derivatives as antileishmanial compounds.
Arch Pharm (Weinheim);
353(8): e1900325, 2020 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-32484266
5.
Synthesis, bioactivity and molecular modeling studies on potential anti-Alzheimer piperidinehydrazide-hydrazones.
Bioorg Chem;
87: 888-900, 2019 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-30538051
6.
Antibacterial activity of porphyrin derivatives against multidrug-resistant bacteria.
Pak J Pharm Sci;
32(5(Special)): 2369-2373, 2019 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-31894020
7.
Synthesis, biological evaluation, and docking studies of some 5-chloro-2(3H)-benzoxazolone Mannich bases derivatives as cholinesterase inhibitors.
Arch Pharm (Weinheim);
351(3-4): e1700273, 2018 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-29527733
8.
Multifunctional cholinesterase inhibitors for Alzheimer's disease: Synthesis, biological evaluations, and docking studies of o/p-propoxyphenylsubstituted-1H-benzimidazole derivatives.
Arch Pharm (Weinheim);
2018 Jul 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-29984517
9.
Synthesis and molecular docking studies of some 4-phthalimidobenzenesulfonamide derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors.
J Enzyme Inhib Med Chem;
32(1): 13-19, 2017 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-27766908
10.
Mannich-Benzimidazole Derivatives as Antioxidant and Anticholinesterase Inhibitors: Synthesis, Biological Evaluations, and Molecular Docking Study.
Arch Pharm (Weinheim);
350(7)2017 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-28379621
11.
Synthesis, Biological Evaluation and Molecular Docking Study of Hydrazone-Containing Pyridinium Salts as Cholinesterase Inhibitors.
Chem Pharm Bull (Tokyo);
64(9): 1281-7, 2016.
Artículo
en Inglés
| MEDLINE | ID: mdl-27581632
12.
Synthesis, biological activity and molecular modeling studies on 1H-benzimidazole derivatives as acetylcholinesterase inhibitors.
Bioorg Med Chem;
21(17): 4928-37, 2013 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23891231
13.
Synthesis and antileishmanial activity of novel pyridinium-hydrazone derivatives.
J Enzyme Inhib Med Chem;
28(5): 960-7, 2013 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-22803671
14.
Design, synthesis, in vitro - In vivo biological evaluation of novel thiazolopyrimidine compounds as antileishmanial agent with PTR1 inhibition.
Eur J Med Chem;
247: 115049, 2023 Feb 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-36577215
15.
The antibacterial activity of photodynamic agents against multidrug resistant bacteria causing wound infection.
Photodiagnosis Photodyn Ther;
40: 103066, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35998880
16.
Interaction of (benzylidene-hydrazono)-1,4-dihydropyridines with beta-amyloid, acetylcholine, and butyrylcholine esterases.
Bioorg Med Chem;
18(5): 2049-59, 2010 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20149667
17.
4-[(2E)-2-(4-Chloro-benzyl-idene)hydrazinyl-idene]-1-methyl-1,4-dihydro-pyridine monohydrate.
Acta Crystallogr Sect E Struct Rep Online;
66(Pt 6): o1324-5, 2010 May 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-21579416
18.
Synthesis and antimicrobial activity of some pyridinium salts.
Molecules;
14(12): 5203-15, 2009 Dec 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-20032886
19.
Photodynamic antimicrobial activity of new porphyrin derivatives against methicillin resistant Staphylococcus aureus.
J Microbiol;
56(11): 828-837, 2018 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-30353469
20.
Synthesis and evaluation of pyridinium-hydrazone derivatives as potential antitumoral agents.
Chem Biol Drug Des;
92(1): 1198-1205, 2018 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-29415336