Detalles de la búsqueda
1.
An initiator-free and solvent-free in-situ self-catalyzed crosslinked polymer electrolyte for all-solid-state lithium-metal batteries.
J Colloid Interface Sci;
648: 972-982, 2023 Oct 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37331078
2.
Pyrazole and pyrimidine phenylacylsulfonamides as dual Bcl-2/Bcl-xL antagonists.
Bioorg Med Chem Lett;
22(12): 3951-6, 2012 Jun 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22608393
3.
Identification of a phenylacylsulfonamide series of dual Bcl-2/Bcl-xL antagonists.
Bioorg Med Chem Lett;
22(12): 3946-50, 2012 Jun 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22608961
4.
Design, synthesis and structure-activity relationships of novel biarylamine-based Met kinase inhibitors.
Bioorg Med Chem Lett;
20(9): 2998-3002, 2010 May 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20382527
5.
Vorasidenib (AG-881): A First-in-Class, Brain-Penetrant Dual Inhibitor of Mutant IDH1 and 2 for Treatment of Glioma.
ACS Med Chem Lett;
11(2): 101-107, 2020 Feb 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-32071674
6.
Discovery of brivanib alaninate ((S)-((R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan-2-yl)2-aminopropanoate), a novel prodrug of dual vascular endothelial growth factor receptor-2 and fibroblast growth factor receptor-1 kinase inhibitor (BMS-540215).
J Med Chem;
51(6): 1976-80, 2008 Mar 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-18288793
7.
Synthesis, SAR, and Evaluation of 4-[2,4-Difluoro-5-(cyclopropylcarbamoyl)phenylamino]pyrrolo[2,1-f][1,2,4]triazine-based VEGFR-2 kinase inhibitors.
Bioorg Med Chem Lett;
18(4): 1354-8, 2008 Feb 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-18221875
8.
Discovery of orally active pyrrolopyridine- and aminopyridine-based Met kinase inhibitors.
Bioorg Med Chem Lett;
18(11): 3224-9, 2008 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-18479916
9.
Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase.
Bioorg Med Chem Lett;
18(6): 1945-51, 2008 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-18289854
10.
Discovery and preclinical studies of 5-isopropyl-6-(5-methyl-1,3,4-oxadiazol-2-yl)-N-(2-methyl-1H-pyrrolo[2,3-b]pyridin-5-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine (BMS-645737), an in vivo active potent VEGFR-2 inhibitor.
Bioorg Med Chem Lett;
18(9): 2985-9, 2008 May 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-18395443
11.
Discovery of AG-120 (Ivosidenib): A First-in-Class Mutant IDH1 Inhibitor for the Treatment of IDH1 Mutant Cancers.
ACS Med Chem Lett;
9(4): 300-305, 2018 Apr 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-29670690
12.
Discovery and preclinical studies of (R)-1-(4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5- methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy)propan- 2-ol (BMS-540215), an in vivo active potent VEGFR-2 inhibitor.
J Med Chem;
49(7): 2143-6, 2006 Apr 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-16570908
13.
Design, synthesis, and evaluation of orally active 4-(2,4-difluoro-5-(methoxycarbamoyl)phenylamino)pyrrolo[2,1-f][1,2,4]triazines as dual vascular endothelial growth factor receptor-2 and fibroblast growth factor receptor-1 inhibitors.
J Med Chem;
48(12): 3991-4008, 2005 Jun 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-15943473
14.
Discovery of aminothiazole inhibitors of cyclin-dependent kinase 2: synthesis, X-ray crystallographic analysis, and biological activities.
J Med Chem;
45(18): 3905-27, 2002 Aug 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-12190313
15.
The antiangiogenic activity in xenograft models of brivanib, a dual inhibitor of vascular endothelial growth factor receptor-2 and fibroblast growth factor receptor-1 kinases.
Mol Cancer Ther;
9(2): 369-78, 2010 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-20103604
16.
Discovery of N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide (BMS-777607), a selective and orally efficacious inhibitor of the Met kinase superfamily.
J Med Chem;
52(5): 1251-4, 2009 Mar 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-19260711
17.
Discovery of pyrrolopyridine-pyridone based inhibitors of Met kinase: synthesis, X-ray crystallographic analysis, and biological activities.
J Med Chem;
51(17): 5330-41, 2008 Sep 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-18690676
18.
Addition of benzylic and allylic organozinc and Grignard reagents to resin-bound imines to provide alpha-branched secondary amines bearing a wide variety of functional groups. Utility in the synthesis of beta-3 adrenergic receptor agonists.
J Comb Chem;
7(1): 99-108, 2005.
Artículo
en Inglés
| MEDLINE | ID: mdl-15638488
19.
Synthesis and SAR of 4-(3-hydroxyphenylamino)pyrrolo[2,1-f][1,2,4]triazine based VEGFR-2 kinase inhibitors.
Bioorg Med Chem Lett;
15(5): 1429-33, 2005 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-15713401
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