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1.
Tonantzitlolone B Modulates the Endogenous Opioid System to Promote Antinociception in Mice.
J Nat Prod;
86(11): 2514-2521, 2023 11 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-37948340
2.
Druggable hot spots in trypanothione reductase: novel insights and opportunities for drug discovery revealed by DRUGpy.
J Comput Aided Mol Des;
35(8): 871-882, 2021 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-34181199
3.
Synthesis and biological evaluation of thiazolidinedione derivatives with high ligand efficiency to P. aeruginosa PhzS.
J Enzyme Inhib Med Chem;
36(1): 1217-1229, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34080514
4.
5-O-methylcneorumchromone K Exerts Antinociceptive Effects in Mice via Interaction with GABAA Receptors.
Int J Mol Sci;
22(7)2021 Mar 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-33810317
5.
Calycopterin, a major flavonoid from Marcetia latifolia, modulates virulence-related traits in Pseudomonas aeruginosa.
Microb Pathog;
144: 104142, 2020 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-32173496
6.
Antileishmanial activity evaluation of thiazolidine-2,4-dione against Leishmania infantum and Leishmania braziliensis.
Parasitol Res;
119(7): 2263-2274, 2020 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-32462293
7.
Dual and selective inhibitors of pteridine reductase 1 (PTR1) and dihydrofolate reductase-thymidylate synthase (DHFR-TS) from Leishmania chagasi.
J Enzyme Inhib Med Chem;
34(1): 1439-1450, 2019 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-31409157
8.
Synthesis and biological evaluation of thiazole derivatives as LbSOD inhibitors.
J Enzyme Inhib Med Chem;
34(1): 333-342, 2019 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-30734600
9.
Quantitative insights towards the design of potent deazaxanthine antagonists of adenosine 2B receptors.
J Enzyme Inhib Med Chem;
29(4): 590-8, 2014 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-24090420
10.
Analysis of the ergosterol biosynthesis pathway cloning, molecular characterization and phylogeny of lanosterol 14 α-demethylase (ERG11) gene of Moniliophthora perniciosa.
Genet Mol Biol;
37(4): 683-93, 2014 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-25505843
11.
DHODH Hot Spots: An Underexplored Source to Guide Drug Development Efforts.
Curr Top Med Chem;
21(23): 2134-2154, 2021.
Artículo
en Inglés
| MEDLINE | ID: mdl-34348625
12.
Triazol-phenyl Antipyretic Derivatives Inhibit mPGES-1 mRNA Levels in LPS-Induced RAW 264.7 Macrophage Cells.
Antiinflamm Antiallergy Agents Med Chem;
20(3): 271-281, 2021.
Artículo
en Inglés
| MEDLINE | ID: mdl-33292158
13.
Adenosine binding to low-molecular-weight purine nucleoside phosphorylase: the structural basis for recognition based on its complex with the enzyme from Schistosoma mansoni.
Acta Crystallogr D Biol Crystallogr;
66(Pt 1): 73-9, 2010 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-20057051
14.
A novel scaffold to fight Pseudomonas aeruginosa pyocyanin production: early steps to novel antivirulence drugs.
Future Med Chem;
12(16): 1489-1503, 2020 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-32772556
15.
Inhibition of intracellular Ca2+ mobilization and potassium channels activation are involved in the vasorelaxation induced by 7-hydroxycoumarin.
Eur J Pharmacol;
887: 173525, 2020 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-32889064
16.
Identification, Characterization and Molecular Modelling Studies of Schistosoma mansoni Dihydrofolate Reductase Inhibitors: From Assay Development to Hit Identification.
Curr Top Med Chem;
18(5): 406-417, 2018.
Artículo
en Inglés
| MEDLINE | ID: mdl-29741139
17.
In vitro and in silico studies of 3-hydroxy-3-methyl-glutaryl coenzyme A reductase inhibitory activity of the cowpea Gln-Asp-Phe peptide.
Food Chem;
259: 270-277, 2018 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-29680054
18.
Nanomolar anti-sickling compounds identified by ligand-based pharmacophore approach.
Eur J Med Chem;
136: 487-496, 2017 Aug 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-28528302
19.
Virtual screening and biological evaluation of novel antipyretic compounds.
Chem Biol Drug Des;
90(5): 739-752, 2017 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-28390086
20.
An integrated approach towards the discovery of novel non-nucleoside Leishmania major pteridine reductase 1 inhibitors.
Eur J Med Chem;
132: 322-332, 2017 May 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-28407565