Detalles de la búsqueda
1.
Alpha-glucosidase inhibitory and hypoglycemic effects of imidazole-bearing thioquinoline derivatives with different substituents: In silico, in vitro, and in vivo evaluations.
Bioorg Chem;
144: 107106, 2024 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-38244380
2.
New 4-phenylpiperazine-carbodithioate-N-phenylacetamide hybrids: Synthesis, in vitro and in silico evaluations against cholinesterase and α-glucosidase enzymes.
Arch Pharm (Weinheim);
355(5): e2100313, 2022 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-35132681
3.
Synthesis, in vitro potency of inhibition, enzyme kinetics and in silico studies of quinoline-based α-glucosidase inhibitors.
Sci Rep;
14(1): 501, 2024 01 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-38177164
4.
Copper supported modified magnetic carrageenan as a bio-based catalyst for the synthesis of novel scaffolds bearing the 1,2,3-triazole unit through the click reaction.
Nanoscale Adv;
6(9): 2337-2349, 2024 Apr 30.
Artículo
en Inglés
| MEDLINE | ID: mdl-38694460
5.
Aryl-quinoline-4-carbonyl hydrazone bearing different 2-methoxyphenoxyacetamides as potent α-glucosidase inhibitors; molecular dynamics, kinetic and structure-activity relationship studies.
Sci Rep;
14(1): 388, 2024 01 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-38172167
6.
Evaluation of novel 2-(quinoline-2-ylthio)acetamide derivatives linked to diphenyl-imidazole as α-glucosidase inhibitors: Insights from in silico, in vitro, and in vivo studies on their anti-diabetic properties.
Eur J Med Chem;
269: 116332, 2024 Apr 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-38508120
7.
Environmentally friendly catalyst- and solvent-free synthesis of 2-anilino nicotinic acids derivatives as potential lead COX inhibitors.
BMC Chem;
17(1): 160, 2023 Nov 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-37986120
8.
Thioquinoline derivatives conjugated to thiosemicarbazide as potent tyrosinase inhibitors with anti-melanogenesis properties.
Sci Rep;
13(1): 2578, 2023 02 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-36782003
9.
Synthesis, ADMT prediction, and in vitro and in silico α-glucosidase inhibition evaluations of new quinoline-quinazolinone-thioacetamides.
RSC Adv;
13(28): 19243-19256, 2023 Jun 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-37377867
10.
New thioxothiazolidinyl-acetamides derivatives as potent urease inhibitors: design, synthesis, in vitro inhibition, and molecular dynamic simulation.
Sci Rep;
13(1): 21, 2023 01 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-36593349
11.
Synthesis, in vitro inhibitor screening, structure-activity relationship, and molecular dynamic simulation studies of novel thioquinoline derivatives as potent α-glucosidase inhibitors.
Sci Rep;
13(1): 7819, 2023 05 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37188744
12.
Synthesis and structure-activity relationship studies of benzimidazole-thioquinoline derivatives as α-glucosidase inhibitors.
Sci Rep;
13(1): 4392, 2023 03 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-36928433
13.
Synthesis and tyrosinase inhibitory activities of novel isopropylquinazolinones.
BMC Chem;
17(1): 65, 2023 Jun 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-37353836
14.
[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole derivatives as new therapeutic candidates against urease positive microorganisms: design, synthesis, pharmacological evaluations, and in silico studies.
Sci Rep;
13(1): 10136, 2023 06 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-37349372
15.
Phenyl-quinoline derivatives as lead structure of cholinesterase inhibitors with potency to reduce the GSK-3ß level targeting Alzheimer's disease.
Int J Biol Macromol;
253(Pt 7): 127392, 2023 Dec 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-37827412
16.
Synthesis and bioactivities evaluation of quinazolin-4(3H)-one derivatives as α-glucosidase inhibitors.
BMC Chem;
16(1): 97, 2022 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-36380337
17.
Design, synthesis, and in silico studies of quinoline-based-benzo[d]imidazole bearing different acetamide derivatives as potent α-glucosidase inhibitors.
Sci Rep;
12(1): 14019, 2022 08 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-35982225
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