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1.

The discovery and evaluation of [¹⁸F]BMS-986229, a novel macrocyclic peptide PET radioligand for the measurement of PD-L1 expression and in-vivo PD-L1 target engagement.

Donnelly, David J; Kim, Joonyoung; Tran, Tritin; Scola, Paul M; Tenney, Daniel; Pena, Adrienne; Petrone, Thomas; Zhang, Yunhui; Boy, Kenneth M; Poss, Michael A; Cole, Erin L; Soars, Matthew G; Johnson, Benjamin M; Cohen, Daniel; Batalla, Daniel; Chow, Patrick L; Shorts, Andrea Olga; Du, Shuyan; Meanwell, Nicholas A; Bonacorsi, Samuel J.

Eur J Nucl Med Mol Imaging; 51(4): 978-990, 2024 Mar.

Artículo en Inglés | MEDLINE | ID: mdl-38049658

2.

Nucleophilic (Radio)Fluorination of Redox-Active Esters via Radical-Polar Crossover Enabled by Photoredox Catalysis.

Webb, Eric W; Park, John B; Cole, Erin L; Donnelly, David J; Bonacorsi, Samuel J; Ewing, William R; Doyle, Abigail G.

J Am Chem Soc; 142(20): 9493-9500, 2020 05 20.

Artículo en Inglés | MEDLINE | ID: mdl-32378889

3.

Chemoselective Methionine Bioconjugation: Site-Selective Fluorine-18 Labeling of Proteins and Peptides.

Lin, Daniel; Wallace, Michael; Allentoff, Alban J; Donnelly, David J; Gomes, Erin; Voronin, Kim; Gong, Sharon; Huang, Richard Y-C; Kim, Ho; Caceres-Cortes, Janet; Bonacorsi, Samuel.

Bioconjug Chem; 31(8): 1908-1916, 2020 08 19.

Artículo en Inglés | MEDLINE | ID: mdl-32687313

4.

Radiosynthesis and preclinical PET evaluation of ⁸⁹Zr-nivolumab (BMS-936558) in healthy non-human primates.

Cole, Erin L; Kim, Joonyoung; Donnelly, David J; Smith, R Adam; Cohen, Daniel; Lafont, Virginie; Morin, Paul E; Huang, Richard Y-C; Chow, Patrick L; Hayes, Wendy; Bonacorsi, Samuel.

Bioorg Med Chem; 25(20): 5407-5414, 2017 Oct 15.

Artículo en Inglés | MEDLINE | ID: mdl-28803798

5.

Synthesis of Diverse (11)C-Labeled PET Radiotracers via Direct Incorporation of [(11)C]CO2.

Mossine, Andrew V; Brooks, Allen F; Jackson, Isaac M; Quesada, Carole A; Sherman, Phillip; Cole, Erin L; Donnelly, David J; Scott, Peter J H; Shao, Xia.

Bioconjug Chem; 27(5): 1382-9, 2016 05 18.

Artículo en Inglés | MEDLINE | ID: mdl-27043721

6.

Development, Characterization, and Radiation Dosimetry Studies of ¹⁸F-BMS-986229, a ¹⁸F-Labeled PD-L1 Macrocyclic Peptide PET Tracer.

Kim, Joonyoung; Donnelly, David J; Tran, Tritin; Pena, Adrienne; Shorts, Andrea Olga; Petrone, Thomas V; Zhang, Yunhui; Boy, Kenneth M; Scola, Paul M; Tenney, Daniel J; Poss, Michael A; Soars, Matthew G; Bonacorsi, Samuel J; Cole, Erin L; Grootendorst, Diederik J; Chow, Patrick L; Meanwell, Nicholas A; Du, Shuyan.

Mol Imaging Biol; 26(2): 301-309, 2024 Apr.

Artículo en Inglés | MEDLINE | ID: mdl-38123744

7.

Transcriptome-wide comparison of sequence variation in divergent ecotypes of kokanee salmon.

Lemay, Matthew A; Donnelly, David J; Russello, Michael A.

BMC Genomics; 14: 308, 2013 May 07.

Artículo en Inglés | MEDLINE | ID: mdl-23651561

8.

Synthesis and Preclinical Evaluation of a ⁶⁸Ga-Labeled Adnectin, ⁶⁸Ga-BMS-986192, as a PET Agent for Imaging PD-L1 Expression.

Robu, Stephanie; Richter, Antonia; Gosmann, Dario; Seidl, Christof; Leung, David; Hayes, Wendy; Cohen, Daniel; Morin, Paul; Donnelly, David J; Lipovsek, Dasa; Bonacorsi, Samuel J; Smith, Adam; Steiger, Katja; Aulehner, Christina; Krackhardt, Angela M; Weber, Wolfgang A.

J Nucl Med; 62(9): 1228-1234, 2021 09 01.

Artículo en Inglés | MEDLINE | ID: mdl-33517324

9.

Evaluation of the Lysophosphatidic Acid Receptor Type 1 Radioligand ¹¹C-BMT-136088 for Lung Imaging in Rhesus Monkeys.

Gallezot, Jean-Dominique; Nabulsi, Nabeel B; Holden, Daniel; Lin, Shu-Fei; Labaree, David; Ropchan, Jim; Najafzadeh, Soheila; Donnelly, David J; Cao, Kai; Bonacorsi, Samuel; Seiders, Jon; Roppe, Jeffrey; Hayes, Wendy; Huang, Yiyun; Du, Shuyan; Carson, Richard E.

J Nucl Med; 59(2): 327-333, 2018 02.

Artículo en Inglés | MEDLINE | ID: mdl-28864634

10.

Synthesis and Biologic Evaluation of a Novel ¹⁸F-Labeled Adnectin as a PET Radioligand for Imaging PD-L1 Expression.

Donnelly, David J; Smith, R Adam; Morin, Paul; Lipovsek, Dasa; Gokemeijer, Jochem; Cohen, Daniel; Lafont, Virginie; Tran, Tritin; Cole, Erin L; Wright, Martin; Kim, Joonyoung; Pena, Adrienne; Kukral, Daniel; Dischino, Douglas D; Chow, Patrick; Gan, Jinping; Adelakun, Olufemi; Wang, Xi-Tao; Cao, Kai; Leung, David; Bonacorsi, Samuel J; Hayes, Wendy.

J Nucl Med; 59(3): 529-535, 2018 03.

Artículo en Inglés | MEDLINE | ID: mdl-29025984

11.

Small Molecule PET Tracers in Drug Discovery.

Donnelly, David J.

Semin Nucl Med; 47(5): 454-460, 2017 09.

Artículo en Inglés | MEDLINE | ID: mdl-28826520

12.

Use of a red cell band 3-ligand/antioxidant to improve red cell storage properties following virucidal phototeatment with chalcogenoxanthylium photosensitizers.

Wagner, Stephen J; Skripchenko, Andrey; Thompson-Montgomery, Dedeene; Awatefe, Helen; Donnelly, David J; Detty, Michael R.

Photochem Photobiol; 82(6): 1595-600, 2006.

Artículo en Inglés | MEDLINE | ID: mdl-16939364

13.

Applications of Fluorine in Medicinal Chemistry.

Gillis, Eric P; Eastman, Kyle J; Hill, Matthew D; Donnelly, David J; Meanwell, Nicholas A.

J Med Chem; 58(21): 8315-59, 2015 Nov 12.

Artículo en Inglés | MEDLINE | ID: mdl-26200936

14.

ATP occlusion by P-glycoprotein as a surrogate measure for drug coupling.

Tombline, Gregory; Holt, Jason J; Gannon, Michael K; Donnelly, David J; Wetzel, Bryan; Sawada, Geri A; Raub, Thomas J; Detty, Michael R.

Biochemistry; 47(10): 3294-307, 2008 Mar 11.

Artículo en Inglés | MEDLINE | ID: mdl-18275155

15.

Stimulation of P-glycoprotein ATPase by analogues of tetramethylrosamine: coupling of drug binding at the "R" site to the ATP hydrolysis transition state.

Tombline, Gregory; Donnelly, David J; Holt, Jason J; You, Youngjae; Ye, Mao; Gannon, Michael K; Nygren, Cara L; Detty, Michael R.

Biochemistry; 45(26): 8034-47, 2006 Jul 04.

Artículo en Inglés | MEDLINE | ID: mdl-16800628

16.

Chalcogenoxanthylium photosensitizers for the photodynamic purging of blood-borne viral and bacterial pathogens.

Wagner, Stephen J; Skripchenko, Andrey; Donnelly, David J; Ramaswamy, Krishna; Detty, Michael R.

Bioorg Med Chem; 13(21): 5927-35, 2005 Nov 01.

Artículo en Inglés | MEDLINE | ID: mdl-16140537

17.

Structure-activity studies of uptake and phototoxicity with heavy-chalcogen analogues of tetramethylrosamine in vitro in chemosensitive and multidrug-resistant cells.

Gibson, Scott L; Holt, Jason J; Ye, Mao; Donnelly, David J; Ohulchanskyy, Tymish Y; You, Youngjae; Detty, Michael R.

Bioorg Med Chem; 13(23): 6394-403, 2005 Dec 01.

Artículo en Inglés | MEDLINE | ID: mdl-16084725

18.

Selenoxanthones via directed metalations in 2-arylselenobenzamide derivatives.

Brennan, Nancy K; Donnelly, David J; Detty, Michael R.

J Org Chem; 68(8): 3344-7, 2003 Apr 18.

Artículo en Inglés | MEDLINE | ID: mdl-12688818

19.

Analogues of tetramethylrosamine as transport molecules for and inhibitors of P-glycoprotein-mediated multidrug resistance.

Gibson, Scott L; Hilf, Russell; Donnelly, David J; Detty, Michael R.

Bioorg Med Chem; 12(17): 4625-31, 2004 Sep 01.

Artículo en Inglés | MEDLINE | ID: mdl-15358289

20.

Synthesis, properties, and photodynamic properties in vitro of heavy-chalcogen analogues of tetramethylrosamine.

Detty, Michael R; Prasad, Paras N; Donnelly, David J; Ohulchanskyy, Tymish; Gibson, Scott L; Hilf, Russell.

Bioorg Med Chem; 12(10): 2537-44, 2004 May 15.

Artículo en Inglés | MEDLINE | ID: mdl-15110836

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