Detalles de la búsqueda
1.
Synthesis, characterization, and biological study of new synthetic opioid hemorphin-4 peptides containing sterically restricted nonnatural amino acids.
Arch Pharm (Weinheim);
: e2400052, 2024 Apr 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-38578075
2.
Synthesis of 2,6-Dimethyltyrosine-Like Amino Acids through Pinacolinamide-Enabled C-H Dimethylation of 4-Dibenzylamino Phenylalanine.
J Org Chem;
87(5): 2580-2589, 2022 03 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-35138099
3.
Identification of small-molecule urea derivatives as PTPC modulators targeting the c subunit of F1/Fo-ATP synthase.
Bioorg Med Chem Lett;
72: 128822, 2022 09 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-35636649
4.
Synthesis and biological evaluation of novel rhodanine-based structures with antiviral activity towards HHV-6 virus.
Bioorg Chem;
119: 105518, 2022 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-34861628
5.
Synthesis and NLRP3-Inflammasome Inhibitory Activity of the Naturally Occurring Velutone F and of Its Non-Natural Regioisomeric Chalconoids.
Int J Mol Sci;
23(16)2022 Aug 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-36012241
6.
In Vivo Bio-Activation of JWH-175 to JWH-018: Pharmacodynamic and Pharmacokinetic Studies in Mice.
Int J Mol Sci;
23(14)2022 Jul 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-35887377
7.
In Vitro and In Vivo Pharmaco-Toxicological Characterization of 1-Cyclohexyl-x-methoxybenzene Derivatives in Mice: Comparison with Tramadol and PCP.
Int J Mol Sci;
22(14)2021 Jul 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-34299276
8.
Worsening of the Toxic Effects of (±)Cis-4,4'-DMAR Following Its Co-Administration with (±)Trans-4,4'-DMAR: Neuro-Behavioural, Physiological, Immunohistochemical and Metabolic Studies in Mice.
Int J Mol Sci;
22(16)2021 Aug 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-34445476
9.
Synthesis and Characterization of Manganese Dithiocarbamate Complexes: New Evidence of Dioxygen Activation.
Molecules;
26(19)2021 Sep 30.
Artículo
en Inglés
| MEDLINE | ID: mdl-34641499
10.
Tetrabranched Hetero-Conjugated Peptides as Bifunctional Agonists of the NOP and Mu Opioid Receptors.
Bioconjug Chem;
30(9): 2444-2451, 2019 09 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-31461266
11.
Biochemically Controlled Release of Dexamethasone Covalently Bound to PEDOT.
Chemistry;
24(41): 10300-10305, 2018 Jul 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-29799647
12.
1-cyclohexyl-x-methoxybenzene derivatives, novel psychoactive substances seized on the internet market. Synthesis and in vivo pharmacological studies in mice.
Hum Psychopharmacol;
32(3)2017 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-28657178
13.
Naphthoquinone amino acid derivatives, synthesis and biological activity as proteasome inhibitors.
J Enzyme Inhib Med Chem;
32(1): 865-877, 2017 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-28657369
14.
Methyl-Containing Pharmaceuticals.
Pharmaceuticals (Basel);
17(5)2024 Apr 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-38794133
15.
Spiropiperidine-Based Oligomycin-Analog Ligands To Counteract the Ischemia-Reperfusion Injury in a Renal Cell Model.
J Med Chem;
67(1): 586-602, 2024 Jan 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-37991993
16.
(L)-Monomethyl Tyrosine (Mmt): New Synthetic Strategy via Bulky 'Forced-Traceless' Regioselective Pd-Catalyzed C(sp2)-H Activation.
Pharmaceuticals (Basel);
16(11)2023 Nov 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-38004457
17.
Dihydroartemisinin-Ursodeoxycholic Bile Acid Hybrids in the Fight against SARS-CoV-2.
ACS Omega;
8(47): 45078-45087, 2023 Nov 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-38046338
18.
In vitro and in vivo pharmaco-dynamic study of the novel fentanyl derivatives: Acrylfentanyl, Ocfentanyl and Furanylfentanyl.
Neuropharmacology;
209: 109020, 2022 05 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-35247453
19.
Structure-Activity Relationship Studies on Oxazolo[3,4-a]pyrazine Derivatives Leading to the Discovery of a Novel Neuropeptide S Receptor Antagonist with Potent In Vivo Activity.
J Med Chem;
64(7): 4089-4108, 2021 04 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-33733768
20.
The Fascinating Chemistry of α-Haloamides.
ChemistryOpen;
9(2): 100-170, 2020 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-32025460