Detalles de la búsqueda
1.
Design, synthesis and biological evaluation of novel quinazoline derivatives as immune checkpoint inhibitors.
Bioorg Med Chem Lett;
108: 129796, 2024 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-38754563
2.
Syntheses and antitumor activities of neorautenol and shinpterocarpin analogs.
Bioorg Med Chem Lett;
91: 129353, 2023 07 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37271378
3.
Design, synthesis and evaluation the bioactivities of novel 1,3-dimethyl-6-amino-1H-indazole derivatives as anticancer agents.
Bioorg Med Chem;
90: 117377, 2023 07 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37352576
4.
Investigation of B,C-ring truncated deguelin derivatives as heat shock protein 90 (HSP90) inhibitors for use as anti-breast cancer agents.
Bioorg Med Chem;
27(7): 1370-1381, 2019 04 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30827868
5.
Potent human glutaminyl cyclase inhibitors as potential anti-Alzheimer's agents: Structure-activity relationship study of Arg-mimetic region.
Bioorg Med Chem;
26(5): 1035-1049, 2018 03 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-29398442
6.
Structure-activity relationship investigation of Phe-Arg mimetic region of human glutaminyl cyclase inhibitors.
Bioorg Med Chem;
26(12): 3133-3144, 2018 07 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-29705377
7.
α-Substituted 2-(3-fluoro-4-methylsulfonamidophenyl)acetamides as potent TRPV1 antagonists.
Bioorg Med Chem Lett;
25(11): 2326-30, 2015 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25937016
8.
α-Methylated simplified resiniferatoxin (sRTX) thiourea analogues as potent and stereospecific TRPV1 antagonists.
Bioorg Med Chem Lett;
24(12): 2685-8, 2014 Jun 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-24794110
9.
2-Aryl substituted pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides as highly potent TRPV1 antagonists.
Bioorg Med Chem Lett;
24(16): 4044-7, 2014 Aug 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-25011915
10.
The HSP90 inhibitor HVH-2930 exhibits potent efficacy against trastuzumab-resistant HER2-positive breast cancer.
Theranostics;
14(6): 2442-2463, 2024.
Artículo
en Inglés
| MEDLINE | ID: mdl-38646654
11.
Structure-activity relationship of human glutaminyl cyclase inhibitors having an N-(5-methyl-1H-imidazol-1-yl)propyl thiourea template.
Bioorg Med Chem;
21(13): 3821-30, 2013 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23643900
12.
TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides.
Bioorg Med Chem;
21(21): 6657-64, 2013 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-24035514
13.
Identifying Possible AChE Inhibitors from Drug-like Molecules via Machine Learning and Experimental Studies.
ACS Omega;
7(24): 20673-20682, 2022 Jun 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-35755364
14.
Discovery of potent indazole-based human glutaminyl cyclase (QC) inhibitors as Anti-Alzheimer's disease agents.
Eur J Med Chem;
244: 114837, 2022 Dec 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-36265279
15.
A novel HSP90 inhibitor SL-145 suppresses metastatic triple-negative breast cancer without triggering the heat shock response.
Oncogene;
41(23): 3289-3297, 2022 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-35501463
16.
Discovery of highly potent human glutaminyl cyclase (QC) inhibitors as anti-Alzheimer's agents by the combination of pharmacophore-based and structure-based design.
Eur J Med Chem;
226: 113819, 2021 Dec 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34536669
17.
Design, synthesis and bioevaluation of novel 6-substituted aminoindazole derivatives as anticancer agents.
RSC Adv;
10(73): 45199-45206, 2020 Dec 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-35516257
18.
In vitro and in silico determination of glutaminyl cyclase inhibitors.
RSC Adv;
9(51): 29619-29627, 2019 Sep 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-35531555
19.
C-terminal HSP90 inhibitor L80 elicits anti-metastatic effects in triple-negative breast cancer via STAT3 inhibition.
Cancer Lett;
447: 141-153, 2019 04 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-30703411
20.
Discovery of Conformationally Restricted Human Glutaminyl Cyclase Inhibitors as Potent Anti-Alzheimer's Agents by Structure-Based Design.
J Med Chem;
62(17): 8011-8027, 2019 09 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-31411468