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1.

Discovery and characterization of bromodomain 2-specific inhibitors of BRDT.

Yu, Zhifeng; Ku, Angela F; Anglin, Justin L; Sharma, Rajesh; Ucisik, Melek Nihan; Faver, John C; Li, Feng; Nyshadham, Pranavanand; Simmons, Nicholas; Sharma, Kiran L; Nagarajan, Sureshbabu; Riehle, Kevin; Kaur, Gundeep; Sankaran, Banumathi; Storl-Desmond, Marta; Palmer, Stephen S; Young, Damian W; Kim, Choel; Matzuk, Martin M.

Proc Natl Acad Sci U S A; 118(9)2021 03 02.

Artículo en Inglés | MEDLINE | ID: mdl-33637650

2.

C-N Coupling of DNA-Conjugated (Hetero)aryl Bromides and Chlorides for DNA-Encoded Chemical Library Synthesis.

Chen, Ying-Chu; Faver, John C; Ku, Angela F; Miklossy, Gabriella; Riehle, Kevin; Bohren, Kurt M; Ucisik, Melek N; Matzuk, Martin M; Yu, Zhifeng; Simmons, Nicholas.

Bioconjug Chem; 31(3): 770-780, 2020 03 18.

Artículo en Inglés | MEDLINE | ID: mdl-32019312

3.

Mycophenolic anilides as broad specificity inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitors.

Lee, Seungheon; Ku, Angela F; Vippila, Mohana Rao; Wang, Yong; Zhang, Minjia; Wang, Xingyou; Hedstrom, Lizbeth; Cuny, Gregory D.

Bioorg Med Chem Lett; 30(24): 127543, 2020 12 15.

Artículo en Inglés | MEDLINE | ID: mdl-32931912

4.

Access to 6a-Alkyl Aporphines: Synthesis of (±)-N-Methylguattescidine.

Ku, Angela F; Cuny, Gregory D.

J Org Chem; 81(20): 10062-10070, 2016 10 21.

Artículo en Inglés | MEDLINE | ID: mdl-27689544

5.

Reversible male contraception by targeted inhibition of serine/threonine kinase 33.

Ku, Angela F; Sharma, Kiran L; Ta, Hai Minh; Sutton, Courtney M; Bohren, Kurt M; Wang, Yong; Chamakuri, Srinivas; Chen, Ruihong; Hakenjos, John M; Jimmidi, Ravikumar; Kent, Katarzyna; Li, Feng; Li, Jian-Yuan; Ma, Lang; Madasu, Chandrashekhar; Palaniappan, Murugesan; Palmer, Stephen S; Qin, Xuan; Robers, Matthew B; Sankaran, Banumathi; Tan, Zhi; Vasquez, Yasmin M; Wang, Jian; Wilkinson, Jennifer; Yu, Zhifeng; Ye, Qiuji; Young, Damian W; Teng, Mingxing; Kim, Choel; Matzuk, Martin M.

Science; 384(6698): 885-890, 2024 May 24.

Artículo en Inglés | MEDLINE | ID: mdl-38781365

6.

Discovery of Highly Potent and BMPR2-Selective Kinase Inhibitors Using DNA-Encoded Chemical Library Screening.

Modukuri, Ram K; Monsivais, Diana; Li, Feng; Palaniappan, Murugesan; Bohren, Kurt M; Tan, Zhi; Ku, Angela F; Wang, Yong; Madasu, Chandrashekhar; Li, Jian-Yuan; Tang, Suni; Miklossy, Gabriella; Palmer, Stephen S; Young, Damian W; Matzuk, Martin M.

J Med Chem; 66(3): 2143-2160, 2023 02 09.

Artículo en Inglés | MEDLINE | ID: mdl-36719862

7.

Discovery of 7-hydroxyaporphines as conformationally restricted ligands for beta-1 and beta-2 adrenergic receptors.

Ku, Angela F; Cuny, Gregory D.

Medchemcomm; 9(2): 353-356, 2018 Feb 01.

Artículo en Inglés | MEDLINE | ID: mdl-30108929

8.

Synthetic studies of 7-oxygenated aporphine alkaloids: preparation of (-)-oliveroline, (-)-nornuciferidine, and derivatives.

Ku, Angela F; Cuny, Gregory D.

Org Lett; 17(5): 1134-7, 2015 Mar 06.

Artículo en Inglés | MEDLINE | ID: mdl-25710592

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Discovery and characterization of bromodomain 2-specific inhibitors of BRDT.

C-N Coupling of DNA-Conjugated (Hetero)aryl Bromides and Chlorides for DNA-Encoded Chemical Library Synthesis.

Mycophenolic anilides as broad specificity inosine-5'-monophosphate dehydrogenase (IMPDH) inhibitors.

Access to 6a-Alkyl Aporphines: Synthesis of (±)-N-Methylguattescidine.

Reversible male contraception by targeted inhibition of serine/threonine kinase 33.

Discovery of Highly Potent and BMPR2-Selective Kinase Inhibitors Using DNA-Encoded Chemical Library Screening.

Discovery of 7-hydroxyaporphines as conformationally restricted ligands for beta-1 and beta-2 adrenergic receptors.

Synthetic studies of 7-oxygenated aporphine alkaloids: preparation of (-)-oliveroline, (-)-nornuciferidine, and derivatives.