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1.
Discovery of (R)-4-cyclopropyl-7,8-difluoro-5-(4-(trifluoromethyl)phenylsulfonyl)-4,5-dihydro-1H-pyrazolo[4,3-c]quinoline (ELND006) and (R)-4-cyclopropyl-8-fluoro-5-(6-(trifluoromethyl)pyridin-3-ylsulfonyl)-4,5-dihydro-2H-pyrazolo[4,3-c]quinoline (ELND007): metabolically stable γ-secretase Inhibitors that selectively inhibit the production of amyloid-ß over Notch.
J Med Chem;
56(13): 5261-74, 2013 Jul 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-23713656
2.
Amyloid precursor protein selective gamma-secretase inhibitors for treatment of Alzheimer's disease.
Alzheimers Res Ther;
2(6): 36, 2010 Dec 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-21190552
3.
A series of C-terminal amino alcohol dipeptide A beta inhibitors.
Bioorg Med Chem Lett;
12(21): 3051-3, 2002 Nov 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-12372499
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