1.
Bioorg Med Chem Lett
; 13(13): 2231-4, 2003 Jul 07.
Artículo
en Inglés
| MEDLINE
| ID: mdl-12798340
RESUMEN
Starting with a micromolar lead identified from high-throughput screening, a series of pyrazoles were discovered with significantly improved potency on bacterial methionyl-tRNA synthetase and selectivity over human methionyl-tRNA synthetase.