Detalles de la búsqueda
1.
Synthesis and biological evaluation of indane-based fluorescent probes for detection of amyloid-ß aggregates in Alzheimer's disease.
Bioorg Med Chem;
95: 117513, 2023 11 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37931520
2.
Neuropathic pain-alleviating effects of pyrazole-conjugated arylsulfonamides as 5-HT6 receptor antagonists.
Bioorg Med Chem Lett;
27(17): 4146-4149, 2017 09 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28729057
3.
Synthesis and diabetic neuropathic pain-alleviating effects of 2N-(pyrazol-3-yl)methylbenzo[d]isothiazole-1,1-dioxide derivatives.
Bioorg Med Chem;
25(17): 4677-4685, 2017 09 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28720324
4.
Synthesis and evaluation of 6-pyrazoylamido-3N-substituted azabicyclo[3,1,0]hexane derivatives as T-type calcium channel inhibitors for treatment of neuropathic pain.
Bioorg Med Chem;
24(21): 5028-5035, 2016 11 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27591007
5.
Monitoring of Intracellular Tau Aggregation Regulated by OGA/OGT Inhibitors.
Int J Mol Sci;
16(9): 20212-24, 2015 Aug 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-26343633
6.
Synthesis and in vitro evaluation of the antitubercular and antibacterial activity of novel oxazolidinones bearing octahydrocyclopenta[c]pyrrol-2-yl moieties.
Chem Pharm Bull (Tokyo);
62(12): 1214-24, 2014.
Artículo
en Inglés
| MEDLINE | ID: mdl-25297523
7.
Synthesis and antibacterial activities of new piperidine substituted (5R)-[1,2,3]triazolylmethyl and (5R)-[(4-F-[1,2,3]triazolyl)methyl] oxazolidinones.
Bioorg Med Chem Lett;
23(5): 1193-6, 2013 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23385213
8.
Synthesis and the 5-HT6 receptor antagonistic effect of 3-arylsulfonylamino-5,6-dihydro-6-substituted pyrazolo[3,4]pyridinones for neuropathic pain treatment.
Bioorg Med Chem Lett;
23(16): 4696-700, 2013 Aug 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-23820387
9.
Discovery of aryl-biphenyl-2-ylmethylpiperazines as novel scaffolds for 5-HT(7) ligands and role of the aromatic substituents in binding to the target receptor.
Bioorg Med Chem;
21(9): 2568-76, 2013 May 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23541835
10.
Oxazolopyridines and thiazolopyridines as monoamine oxidase B inhibitors for the treatment of Parkinson's disease.
Bioorg Med Chem;
21(17): 5480-7, 2013 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23810676
11.
Synthetic Strategy for Aryl(alkynyl)phosphinates by a Three-Component Coupling Reaction Involving Arynes, Phosphites, and Alkynes.
Org Lett;
24(45): 8295-8299, 2022 Nov 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-36342701
12.
Discovery of piperidinyl aminopyrimidine derivatives as IKK-2 inhibitors.
Bioorg Med Chem Lett;
21(10): 3002-6, 2011 May 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-21489792
13.
Antioxidant Compound, Oxyresveratrol, Inhibits APP Production through the AMPK/ULK1/mTOR-Mediated Autophagy Pathway in Mouse Cortical Astrocytes.
Antioxidants (Basel);
10(3)2021 Mar 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-33800526
14.
"Turn-On" Quinoline-Based Fluorescent Probe for Selective Imaging of Tau Aggregates in Alzheimer's Disease: Rational Design, Synthesis, and Molecular Docking.
ACS Sens;
6(6): 2281-2289, 2021 06 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-34115933
15.
Novel quinoline-based fluorescent bioimaging probe, KSNP117, for sentinel lymph node mapping.
J Mater Chem B;
9(24): 4857-4862, 2021 06 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-34076031
16.
Synthesis and antibacterial activity of new 9-O-arylpropenyloxime ketolides.
Bioorg Med Chem Lett;
20(8): 2671-4, 2010 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20338761
17.
Novel 6-N-arylcarboxamidopyrazolo[4,3-d]pyrimidin-7-one derivatives as potential anti-cancer agents.
Bioorg Med Chem Lett;
20(5): 1630-3, 2010 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20138760
18.
O-GlcNAcase: Emerging Mechanism, Substrate Recognition and Small-Molecule Inhibitors.
ChemMedChem;
15(14): 1244-1257, 2020 07 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-32496638
19.
Quinazolindione derivatives as potent 5-HT3A receptor antagonists.
Bioorg Med Chem;
17(13): 4793-6, 2009 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19447040
20.
Functional human 5-HT6 receptor assay for high throughput screening of chemical ligands and binding proteins.
Comb Chem High Throughput Screen;
11(4): 316-24, 2008 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-18473741