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1.
Emergence of Japanese encephalitis in eastern parts of Madhya Pradesh, India.
J Vector Borne Dis;
60(2): 215-219, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-37417173
2.
Discovery of (R)-(3-fluoropyrrolidin-1-yl)(6-((5-(trifluoromethyl)pyridin-2-yl)oxy)quinolin-2-yl)methanone (ABBV-318) and analogs as small molecule Nav1.7/ Nav1.8 blockers for the treatment of pain.
Bioorg Med Chem;
63: 116743, 2022 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-35436748
3.
Rational design, synthesis, and structure-activity relationships of 5-amino-1H-pyrazole-4-carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors.
Bioorg Med Chem;
25(1): 67-74, 2017 01 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28340988
4.
Anti-TNF Thioester Glucocorticoid Antibody-Drug Conjugate Fully Inhibits Inflammation with Minimal Effect on Systemic Corticosterone Levels in a Mouse Arthritis Model.
J Med Chem;
67(11): 9495-9515, 2024 Jun 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-38780432
5.
Gamma interferon release assay for monitoring of treatment response for active tuberculosis: an explosion in the spaghetti factory.
J Clin Microbiol;
51(2): 607-10, 2013 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-23175268
6.
Discovery of novel and potent heterocyclic carboxylic acid derivatives as protein tyrosine phosphatase 1B inhibitors.
Bioorg Med Chem Lett;
22(8): 2843-9, 2012 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22424978
7.
Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate.
J Med Chem;
65(23): 15893-15934, 2022 12 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-36394224
8.
Innovating the treatment of COPD exacerbations: a phone interactive telesystem to increase COPD Action Plan adherence.
BMJ Open Respir Res;
6(1): e000379, 2019.
Artículo
en Inglés
| MEDLINE | ID: mdl-31178998
9.
Correction to "Discovery of ABBV-3373, an Anti-TNF Glucocorticoid Receptor Modulator Immunology Antibody Drug Conjugate".
J Med Chem;
66(8): 6010, 2023 Apr 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-37027784
10.
Fatty acid amide hydrolase inhibitors display broad selectivity and inhibit multiple carboxylesterases as off-targets.
Neuropharmacology;
52(4): 1095-105, 2007 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-17217969
11.
Discovery of Potent and Selective A2A Antagonists with Efficacy in Animal Models of Parkinson's Disease and Depression.
ACS Med Chem Lett;
8(8): 835-840, 2017 Aug 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-28835798
12.
A2B adenosine receptor antagonists: Design, synthesis and biological evaluation of novel xanthine derivatives.
Eur J Med Chem;
127: 986-996, 2017 Feb 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-27842891
13.
Design and synthesis of novel xanthine derivatives as potent and selective A2B adenosine receptor antagonists for the treatment of chronic inflammatory airway diseases.
Eur J Med Chem;
134: 218-229, 2017 Jul 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-28415011
14.
Design, Synthesis of Novel, Potent, Selective, Orally Bioavailable Adenosine A2A Receptor Antagonists and Their Biological Evaluation.
J Med Chem;
60(2): 681-694, 2017 01 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-28055204
15.
1-aryl-3-(4-pyridine-2-ylpiperazin-1-yl)propan-1-one oximes as potent dopamine D4 receptor agonists for the treatment of erectile dysfunction.
J Med Chem;
49(17): 5093-109, 2006 Aug 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-16913699
16.
Discovery of 3-methyl-N-(1-oxy-3',4',5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-ylmethyl)benzamide (ABT-670), an orally bioavailable dopamine D4 agonist for the treatment of erectile dysfunction.
J Med Chem;
49(25): 7450-65, 2006 Dec 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-17149874
17.
Structure-activity relationship of triazafluorenone derivatives as potent and selective mGluR1 antagonists.
J Med Chem;
48(23): 7374-88, 2005 Nov 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-16279797
18.
A-412997 is a selective dopamine D4 receptor agonist in rats.
Pharmacol Biochem Behav;
82(1): 140-7, 2005 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-16153699
19.
Discovery of 2-(4-pyridin-2-ylpiperazin-1-ylmethyl)-1H-benzimidazole (ABT-724), a dopaminergic agent with a novel mode of action for the potential treatment of erectile dysfunction.
J Med Chem;
47(15): 3853-64, 2004 Jul 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-15239663
20.
Synthesis and structure-activity studies on N-[5-(1H-imidazol-4-yl)-5,6,7,8-tetrahydro-1-naphthalenyl]methanesulfonamide, an imidazole-containing alpha(1A)-adrenoceptor agonist.
J Med Chem;
47(12): 3220-35, 2004 Jun 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-15163201