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1.
PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc.
Int J Mol Sci;
22(23)2021 Dec 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-34884931
2.
Affinity-based separation methods for the study of biological interactions: The case of peroxisome proliferator-activated receptors in drug discovery.
Methods;
146: 12-25, 2018 08 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29462658
3.
Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity.
J Enzyme Inhib Med Chem;
31(sup4): 25-37, 2016.
Artículo
en Inglés
| MEDLINE | ID: mdl-27556138
4.
LT175 is a novel PPARα/γ ligand with potent insulin-sensitizing effects and reduced adipogenic properties.
J Biol Chem;
289(10): 6908-6920, 2014 Mar 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-24451380
5.
Structural basis of the transactivation deficiency of the human PPARγ F360L mutant associated with familial partial lipodystrophy.
Acta Crystallogr D Biol Crystallogr;
70(Pt 7): 1965-76, 2014 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-25004973
6.
Design and biophysical characterization of atrazine-sensing peptides mimicking the Chlamydomonas reinhardtii plastoquinone binding niche.
Phys Chem Chem Phys;
15(31): 13108-15, 2013 Aug 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-23824019
7.
Synthesis, biological evaluation and molecular investigation of fluorinated peroxisome proliferator-activated receptors α/γ dual agonists.
Bioorg Med Chem;
20(6): 2141-51, 2012 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22341573
8.
Cytosolic localization and in vitro assembly of human de novo thymidylate synthesis complex.
FEBS J;
289(6): 1625-1649, 2022 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-34694685
9.
Discovery of Novel Chemical Series of OXA-48 ß-Lactamase Inhibitors by High-Throughput Screening.
Pharmaceuticals (Basel);
14(7)2021 Jun 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-34202402
10.
Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy.
Pharmaceuticals (Basel);
13(6)2020 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-32492898
11.
A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor γ Binding Properties and Biological Activities.
J Med Chem;
63(21): 13124-13139, 2020 11 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-33142057
12.
Insights into PPARγ Phosphorylation and Its Inhibition Mechanism.
J Med Chem;
63(9): 4811-4823, 2020 05 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-32239932
13.
Surface Plasmon Resonance as a Tool for Ligand Binding Investigation of Engineered GPR17 Receptor, a G Protein Coupled Receptor Involved in Myelination.
Front Chem;
7: 910, 2019.
Artículo
en Inglés
| MEDLINE | ID: mdl-31998697
14.
Identification of the First PPARα/γ Dual Agonist Able To Bind to Canonical and Alternative Sites of PPARγ and To Inhibit Its Cdk5-Mediated Phosphorylation.
J Med Chem;
61(18): 8282-8298, 2018 09 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-30199253
15.
Stereoselectivity by enantiomeric inhibitors of matrix metalloproteinase-8: new insights from molecular dynamics simulations.
J Med Chem;
50(2): 211-8, 2007 Jan 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-17228863
16.
Betulinic acid is a PPARγ antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis.
Sci Rep;
7(1): 5777, 2017 07 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-28720829
17.
Structural insight into the stereoselective inhibition of MMP-8 by enantiomeric sulfonamide phosphonates.
J Med Chem;
49(3): 923-31, 2006 Feb 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-16451058
18.
Screening of saponins and sapogenins from Medicago species as potential PPARγ agonists and X-ray structure of the complex PPARγ/caulophyllogenin.
Sci Rep;
6: 27658, 2016 06 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-27283034
19.
Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode.
Sci Rep;
6: 34792, 2016 10 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-27708429
20.
On the metabolically active form of metaglidasen: improved synthesis and investigation of its peculiar activity on peroxisome proliferator-activated receptors and skeletal muscles.
ChemMedChem;
10(3): 555-65, 2015 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-25641779