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1.
Small-molecule inhibitors prevent the genotoxic and protumoural effects induced by colibactin-producing bacteria.
Gut;
65(2): 278-85, 2016 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-25588406
2.
Crystal Structures of KPC-2 and SHV-1 ß-Lactamases in Complex with the Boronic Acid Transition State Analog S02030.
Antimicrob Agents Chemother;
60(3): 1760-6, 2016 Jan 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-26729491
3.
Boronic Acid Transition State Inhibitors Active against KPC and Other Class A ß-Lactamases: Structure-Activity Relationships as a Guide to Inhibitor Design.
Antimicrob Agents Chemother;
60(3): 1751-9, 2016 Jan 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-26729496
4.
Synthesis of 1,2,3-triazol-1-yl-methaneboronic acids via click chemistry: an easy access to a new potential scaffold for protease inhibitors.
European J Org Chem;
2015(5): 1075-1083, 2015 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-26257579
5.
Fragment-guided design of subnanomolar ß-lactamase inhibitors active in vivo.
Proc Natl Acad Sci U S A;
109(43): 17448-53, 2012 Oct 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-23043117
6.
Biochemical and structural analysis of inhibitors targeting the ADC-7 cephalosporinase of Acinetobacter baumannii.
Biochemistry;
53(48): 7670-9, 2014 Dec 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-25380506
7.
Structure-Based Analysis of Boronic Acids as Inhibitors of Acinetobacter-Derived Cephalosporinase-7, a Unique Class C ß-Lactamase.
ACS Infect Dis;
4(3): 325-336, 2018 03 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-29144724
8.
Inhibition of Acinetobacter-Derived Cephalosporinase: Exploring the Carboxylate Recognition Site Using Novel ß-Lactamase Inhibitors.
ACS Infect Dis;
4(3): 337-348, 2018 03 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-29144725
9.
Click Chemistry in Lead Optimization of Boronic Acids as ß-Lactamase Inhibitors.
J Med Chem;
58(14): 5445-58, 2015 Jul 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-26102369
10.
Inhibiting the ß-Lactamase of Mycobacterium tuberculosis (Mtb) with Novel Boronic Acid Transition-State Inhibitors (BATSIs).
ACS Infect Dis;
1(6): 234-42, 2015 Jun 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-27622739
11.
Design and exploration of novel boronic acid inhibitors reveals important interactions with a clavulanic acid-resistant sulfhydryl-variable (SHV) ß-lactamase.
J Med Chem;
56(3): 1084-97, 2013 Feb 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-23252553
12.
Design, synthesis, crystal structures, and antimicrobial activity of sulfonamide boronic acids as ß-lactamase inhibitors.
J Med Chem;
53(21): 7852-63, 2010 Nov 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-20945905
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