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1.
Discovery and optimization of pyrazole amides as antagonists of CCR1.
Bioorg Med Chem Lett;
29(3): 435-440, 2019 02 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30455146
2.
Selective CB2 receptor agonists. Part 1: the identification of novel ligands through computer-aided drug design (CADD) approaches.
Bioorg Med Chem Lett;
25(3): 575-80, 2015 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25556098
3.
Selective CB2 receptor agonists. Part 2: Structure-activity relationship studies and optimization of proline-based compounds.
Bioorg Med Chem Lett;
25(3): 581-6, 2015 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25556092
4.
Selective CB2 receptor agonists. Part 3: the optimization of a piperidine-based series that demonstrated efficacy in an in vivo neuropathic pain model.
Bioorg Med Chem Lett;
25(3): 587-92, 2015 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25575658
5.
Discovery of a potent and dissociated non-steroidal glucocorticoid receptor agonist containing an alkyl carbinol pharmacophore.
Bioorg Med Chem Lett;
24(8): 1934-40, 2014 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-24656565
6.
1,4-Diazepane compounds as potent and selective CB2 agonists: optimization of metabolic stability.
Bioorg Med Chem Lett;
21(7): 2011-6, 2011 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-21354795
7.
Non-steroidal dissociated glucocorticoid agonists: indoles as A-ring mimetics and function-regulating pharmacophores.
Bioorg Med Chem Lett;
21(22): 6842-51, 2011 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-21963986
8.
Quinol-4-ones as steroid A-ring mimetics in nonsteroidal dissociated glucocorticoid agonists.
J Med Chem;
49(26): 7887-96, 2006 Dec 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-17181172
9.
Synthesis, SAR, and series evolution of novel oxadiazole-containing 5-lipoxygenase activating protein inhibitors: discovery of 2-[4-(3-{(r)-1-[4-(2-amino-pyrimidin-5-yl)-phenyl]-1-cyclopropyl-ethyl}-[1,2,4]oxadiazol-5-yl)-pyrazol-1-yl]-N,N-dimethyl-acetamide (BI 665915).
J Med Chem;
58(4): 1669-90, 2015 Feb 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-25671290
10.
Design and synthesis of dipeptide nitriles as reversible and potent Cathepsin S inhibitors.
J Med Chem;
45(25): 5471-82, 2002 Dec 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-12459015
11.
Optimization of drug-like properties of nonsteroidal glucocorticoid mimetics and identification of a clinical candidate.
ACS Med Chem Lett;
5(12): 1318-23, 2014 Dec 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-25516791
12.
Identification of highly efficacious glucocorticoid receptor agonists with a potential for reduced clinical bone side effects.
J Med Chem;
57(4): 1583-98, 2014 Feb 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-24506830
13.
Nonsteroidal dissociated glucocorticoid agonists containing azaindoles as steroid A-ring mimetics.
J Med Chem;
53(18): 6681-98, 2010 Sep 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-20735001
14.
Alpha-methyltryptamine sulfonamide derivatives as novel glucocorticoid receptor ligands.
Bioorg Med Chem Lett;
17(2): 315-9, 2007 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-17118655
15.
Identification of a novel class of succinyl-nitrile-based Cathepsin S inhibitors.
Bioorg Med Chem Lett;
17(9): 2465-9, 2007 May 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-17379516
16.
A concise asymmetric route for the synthesis of a novel class of glucocorticoid mimetics containing a trifluoromethyl-substituted alcohol.
Bioorg Med Chem Lett;
16(3): 654-7, 2006 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-16263276
17.
Trifluoromethyl group as a pharmacophore: effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand.
Bioorg Med Chem Lett;
15(21): 4761-9, 2005 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-16112571
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