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Anilino-monoindolylmaleimides as potent and selective JAK3 inhibitors.
McDonnell, Mark E; Bian, Haiyan; Wrobel, Jay; Smith, Garry R; Liang, Shuguang; Ma, Haiching; Reitz, Allen B.
Afiliación
  • McDonnell ME; Fox Chase Chemical Diversity Center, Inc., 3805 Old Easton Road, Doylestown, PA 18902, United States.
  • Bian H; Fox Chase Chemical Diversity Center, Inc., 3805 Old Easton Road, Doylestown, PA 18902, United States.
  • Wrobel J; Fox Chase Chemical Diversity Center, Inc., 3805 Old Easton Road, Doylestown, PA 18902, United States. Electronic address: jwrobel@fc-cdci.com.
  • Smith GR; Fox Chase Chemical Diversity Center, Inc., 3805 Old Easton Road, Doylestown, PA 18902, United States.
  • Liang S; Reaction Biology, Corp., One Great Valley Parkway, Suite 2, Malvern, PA 19355, United States.
  • Ma H; Reaction Biology, Corp., One Great Valley Parkway, Suite 2, Malvern, PA 19355, United States.
  • Reitz AB; Fox Chase Chemical Diversity Center, Inc., 3805 Old Easton Road, Doylestown, PA 18902, United States.
Bioorg Med Chem Lett ; 24(4): 1116-21, 2014 Feb 15.
Article en En | MEDLINE | ID: mdl-24461299

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Inhibidores de Proteínas Quinasas / Janus Quinasa 3 / Compuestos de Anilina / Maleimidas Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2014 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Inhibidores de Proteínas Quinasas / Janus Quinasa 3 / Compuestos de Anilina / Maleimidas Límite: Humans Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2014 Tipo del documento: Article País de afiliación: Estados Unidos