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Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors.
Jakopin, Ziga; Ilas, Janez; Barancoková, Michaela; Brvar, Matjaz; Tammela, Päivi; Sollner Dolenc, Marija; Tomasic, Tihomir; Kikelj, Danijel.
Afiliación
  • Jakopin Z; University of Ljubljana, Faculty of Pharmacy, Askerceva 7, 1000 Ljubljana, Slovenia. Electronic address: ziga.jakopin@ffa.uni-lj.si.
  • Ilas J; University of Ljubljana, Faculty of Pharmacy, Askerceva 7, 1000 Ljubljana, Slovenia.
  • Barancoková M; University of Ljubljana, Faculty of Pharmacy, Askerceva 7, 1000 Ljubljana, Slovenia.
  • Brvar M; National Institute of Chemistry, Laboratory for Molecular Modeling, Hajdrihova ulica 19, 1001 Ljubljana, Slovenia.
  • Tammela P; University of Helsinki, Faculty of Pharmacy, Division of Pharmaceutical Biosciences, P.O. Box 56, FI-00014 Helsinki, Finland.
  • Sollner Dolenc M; University of Ljubljana, Faculty of Pharmacy, Askerceva 7, 1000 Ljubljana, Slovenia.
  • Tomasic T; University of Ljubljana, Faculty of Pharmacy, Askerceva 7, 1000 Ljubljana, Slovenia.
  • Kikelj D; University of Ljubljana, Faculty of Pharmacy, Askerceva 7, 1000 Ljubljana, Slovenia.
Eur J Med Chem ; 130: 171-184, 2017 Apr 21.
Article en En | MEDLINE | ID: mdl-28246042

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Oxadiazoles / Topoisomerasa de ADN IV / Inhibidores de Topoisomerasa II / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2017 Tipo del documento: Article

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Oxadiazoles / Topoisomerasa de ADN IV / Inhibidores de Topoisomerasa II / Antibacterianos Idioma: En Revista: Eur J Med Chem Año: 2017 Tipo del documento: Article