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GNE-371, a Potent and Selective Chemical Probe for the Second Bromodomains of Human Transcription-Initiation-Factor TFIID Subunit 1 and Transcription-Initiation-Factor TFIID Subunit 1-like.
Wang, Shumei; Tsui, Vickie; Crawford, Terry D; Audia, James E; Burdick, Daniel J; Beresini, Maureen H; Côté, Alexandre; Cummings, Richard; Duplessis, Martin; Flynn, E Megan; Hewitt, Michael C; Huang, Hon-Ren; Jayaram, Hariharan; Jiang, Ying; Joshi, Shivangi; Murray, Jeremy; Nasveschuk, Christopher G; Pardo, Eneida; Poy, Florence; Romero, F Anthony; Tang, Yong; Taylor, Alexander M; Wang, Jian; Xu, Zhaowu; Zawadzke, Laura E; Zhu, Xiaoyu; Albrecht, Brian K; Magnuson, Steven R; Bellon, Steve; Cochran, Andrea G.
Afiliación
  • Wang S; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Tsui V; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Crawford TD; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Audia JE; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Burdick DJ; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Beresini MH; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Cummings R; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Duplessis M; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Flynn EM; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Hewitt MC; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Huang HR; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Jayaram H; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Jiang Y; Wuxi Apptec Company, Ltd. , 288 Fute Zhong Road , Waigaoqiao Free Trade Zone, Shanghai 200131 , People's Republic of China.
  • Joshi S; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Murray J; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Nasveschuk CG; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Pardo E; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Poy F; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Romero FA; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Tang Y; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Taylor AM; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Wang J; Wuxi Apptec Company, Ltd. , 288 Fute Zhong Road , Waigaoqiao Free Trade Zone, Shanghai 200131 , People's Republic of China.
  • Xu Z; Wuxi Apptec Company, Ltd. , 288 Fute Zhong Road , Waigaoqiao Free Trade Zone, Shanghai 200131 , People's Republic of China.
  • Zawadzke LE; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Zhu X; Wuxi Apptec Company, Ltd. , 288 Fute Zhong Road , Waigaoqiao Free Trade Zone, Shanghai 200131 , People's Republic of China.
  • Albrecht BK; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Magnuson SR; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
  • Bellon S; Constellation Pharmaceuticals , 215 First Street, Suite 200 , Cambridge , Massachusetts 02142 , United States.
  • Cochran AG; Genentech Inc. , 1 DNA Way , South San Francisco , California 94080 , United States.
J Med Chem ; 61(20): 9301-9315, 2018 10 25.
Article en En | MEDLINE | ID: mdl-30289257

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Bencimidazoles / Diseño de Fármacos / Sondas Moleculares / Factor de Transcripción TFIID Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Bencimidazoles / Diseño de Fármacos / Sondas Moleculares / Factor de Transcripción TFIID Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2018 Tipo del documento: Article País de afiliación: Estados Unidos