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Design, synthesis and biological evaluation of bifunctional inhibitors of membrane type 1 matrix metalloproteinase (MT1-MMP).
Cuffaro, Doretta; Nuti, Elisa; Gifford, Valentina; Ito, Noriko; Camodeca, Caterina; Tuccinardi, Tiziano; Nencetti, Susanna; Orlandini, Elisabetta; Itoh, Yoshifumi; Rossello, Armando.
Afiliación
  • Cuffaro D; Department of Pharmacy, Università di Pisa, via Bonanno 6, 56126 Pisa, Italy.
  • Nuti E; Department of Pharmacy, Università di Pisa, via Bonanno 6, 56126 Pisa, Italy.
  • Gifford V; Kennedy Institute of Rheumatology, Nuffield Department of Orthopaedics, Rheumatology and Musculoskeletal Sciences, University of Oxford, Oxford OX3 7FY, United Kingdom.
  • Ito N; Kennedy Institute of Rheumatology, Nuffield Department of Orthopaedics, Rheumatology and Musculoskeletal Sciences, University of Oxford, Oxford OX3 7FY, United Kingdom.
  • Camodeca C; Department of Pharmacy, Università di Pisa, via Bonanno 6, 56126 Pisa, Italy.
  • Tuccinardi T; Department of Pharmacy, Università di Pisa, via Bonanno 6, 56126 Pisa, Italy.
  • Nencetti S; Department of Pharmacy, Università di Pisa, via Bonanno 6, 56126 Pisa, Italy.
  • Orlandini E; Department of Earth Sciences, University of Pisa, Via Santa Maria 53, 56126 Pisa, Italy.
  • Itoh Y; Kennedy Institute of Rheumatology, Nuffield Department of Orthopaedics, Rheumatology and Musculoskeletal Sciences, University of Oxford, Oxford OX3 7FY, United Kingdom.
  • Rossello A; Department of Pharmacy, Università di Pisa, via Bonanno 6, 56126 Pisa, Italy. Electronic address: armando.rossello@farm.unipi.it.
Bioorg Med Chem ; 27(1): 196-207, 2019 01 01.
Article en En | MEDLINE | ID: mdl-30522899

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Sulfonamidas / Metaloproteinasa 14 de la Matriz / Inhibidores de la Metaloproteinasa de la Matriz / Ácidos Hidroxámicos Límite: Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Sulfonamidas / Metaloproteinasa 14 de la Matriz / Inhibidores de la Metaloproteinasa de la Matriz / Ácidos Hidroxámicos Límite: Humans Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2019 Tipo del documento: Article País de afiliación: Italia