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Dual targeting of PTP1B and glucosidases with new bifunctional iminosugar inhibitors to address type 2 diabetes.
Ferhati, Xhenti; Matassini, Camilla; Fabbrini, Maria Giulia; Goti, Andrea; Morrone, Amelia; Cardona, Francesca; Moreno-Vargas, Antonio J; Paoli, Paolo.
Afiliación
  • Ferhati X; Department of Chemistry 'Ugo Schiff', University of Firenze, via della Lastruccia 3-13, Sesto Fiorentino, (FI), Italy.
  • Matassini C; Department of Chemistry 'Ugo Schiff', University of Firenze, via della Lastruccia 3-13, Sesto Fiorentino, (FI), Italy.
  • Fabbrini MG; Department of Chemistry 'Ugo Schiff', University of Firenze, via della Lastruccia 3-13, Sesto Fiorentino, (FI), Italy.
  • Goti A; Department of Chemistry 'Ugo Schiff', University of Firenze, via della Lastruccia 3-13, Sesto Fiorentino, (FI), Italy; Associated with Consorzio Interuniversitario Nazionale di ricerca in Metodologie e Processi Innovativi di Sintesi (CINMPIS), Italy.
  • Morrone A; Paediatric Neurology Unit and Laboratories, Neuroscience Department, Meyer Children's Hospital, and Department of Neurosciences, Pharmacology and Child Health. University of Florence, Viale Pieraccini n. 24, 50139 Firenze, Italy.
  • Cardona F; Department of Chemistry 'Ugo Schiff', University of Firenze, via della Lastruccia 3-13, Sesto Fiorentino, (FI), Italy; Associated with Consorzio Interuniversitario Nazionale di ricerca in Metodologie e Processi Innovativi di Sintesi (CINMPIS), Italy. Electronic address: francesca.cardona@unifi.it.
  • Moreno-Vargas AJ; Departamento de Química Orgánica, Facultad de Química, Universidad de Sevilla, n/Prof. García González 1, E-41012 Sevilla, Spain.
  • Paoli P; Department of Experimental and Clinical Biomedical Sciences, University of Florence, Viale Morgagni 50, 50134 Florence, Italy. Electronic address: paolo.paoli@unifi.it.
Bioorg Chem ; 87: 534-549, 2019 06.
Article en En | MEDLINE | ID: mdl-30928876

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Diabetes Mellitus Tipo 2 / Iminoazúcares / Proteína Tirosina Fosfatasa no Receptora Tipo 1 / Glucosidasas / Hipoglucemiantes Límite: Humans Idioma: En Revista: Bioorg Chem Año: 2019 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Diabetes Mellitus Tipo 2 / Iminoazúcares / Proteína Tirosina Fosfatasa no Receptora Tipo 1 / Glucosidasas / Hipoglucemiantes Límite: Humans Idioma: En Revista: Bioorg Chem Año: 2019 Tipo del documento: Article País de afiliación: Italia