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ABC-transporter upregulation mediates resistance to the CDK7 inhibitors THZ1 and ICEC0942.
Sava, Georgina P; Fan, Hailing; Fisher, Rosemary A; Lusvarghi, Sabrina; Pancholi, Sunil; Ambudkar, Suresh V; Martin, Lesley-Ann; Charles Coombes, R; Buluwela, Lakjaya; Ali, Simak.
Afiliación
  • Sava GP; Division of Cancer, Department of Surgery & Cancer, Imperial College London, Hammersmith Hospital Campus, London, UK.
  • Fan H; Division of Cancer, Department of Surgery & Cancer, Imperial College London, Hammersmith Hospital Campus, London, UK.
  • Fisher RA; Division of Cancer, Department of Surgery & Cancer, Imperial College London, Hammersmith Hospital Campus, London, UK.
  • Lusvarghi S; Laboratory of Cell Biology, Center for Cancer Research, National Cancer Institute, Bethesda, MD, 20892, USA.
  • Pancholi S; The Breast Cancer Now Toby Robins Research Centre, The Institute of Cancer Research, London, UK.
  • Ambudkar SV; Laboratory of Cell Biology, Center for Cancer Research, National Cancer Institute, Bethesda, MD, 20892, USA.
  • Martin LA; The Breast Cancer Now Toby Robins Research Centre, The Institute of Cancer Research, London, UK.
  • Charles Coombes R; Division of Cancer, Department of Surgery & Cancer, Imperial College London, Hammersmith Hospital Campus, London, UK.
  • Buluwela L; Division of Cancer, Department of Surgery & Cancer, Imperial College London, Hammersmith Hospital Campus, London, UK.
  • Ali S; Division of Cancer, Department of Surgery & Cancer, Imperial College London, Hammersmith Hospital Campus, London, UK. simak.ali@imperial.ac.uk.
Oncogene ; 39(3): 651-663, 2020 01.
Article en En | MEDLINE | ID: mdl-31530935

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Regulación Neoplásica de la Expresión Génica / Quinasas Ciclina-Dependientes / Resistencia a Antineoplásicos / Inhibidores de Proteínas Quinasas / Transportador de Casetes de Unión a ATP, Subfamilia G, Miembro 2 / Proteínas de Neoplasias Tipo de estudio: Prognostic_studies Límite: Female / Humans Idioma: En Revista: Oncogene Asunto de la revista: BIOLOGIA MOLECULAR / NEOPLASIAS Año: 2020 Tipo del documento: Article País de afiliación: Reino Unido

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Regulación Neoplásica de la Expresión Génica / Quinasas Ciclina-Dependientes / Resistencia a Antineoplásicos / Inhibidores de Proteínas Quinasas / Transportador de Casetes de Unión a ATP, Subfamilia G, Miembro 2 / Proteínas de Neoplasias Tipo de estudio: Prognostic_studies Límite: Female / Humans Idioma: En Revista: Oncogene Asunto de la revista: BIOLOGIA MOLECULAR / NEOPLASIAS Año: 2020 Tipo del documento: Article País de afiliación: Reino Unido