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Novel indolylarylsulfone derivatives as covalent HIV-1 reverse transcriptase inhibitors specifically targeting the drug-resistant mutant Y181C.
Gao, Ping; Song, Shu; Frutos-Beltrán, Estrella; Li, Wenxin; Sun, Bin; Kang, Dongwei; Zou, Jinmi; Zhang, Jian; Pannecouque, Christophe; De Clercq, Erik; Menéndez-Arias, Luis; Zhan, Peng; Liu, Xinyong.
Afiliación
  • Gao P; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China.
  • Song S; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China.
  • Frutos-Beltrán E; Centro de Biología Molecular "Severo Ochoa" (Consejo Superior de Investigaciones Científicas & Universidad Autónoma de Madrid), Madrid, Spain.
  • Li W; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China.
  • Sun B; Institute of BioPharmaceutical Research, Liaocheng University, 1 Hunan Road, Liaocheng 252000, PR China.
  • Kang D; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China.
  • Zou J; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China.
  • Zhang J; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China.
  • Pannecouque C; Rega Institute for Medical Research, K. U. Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium.
  • De Clercq E; Rega Institute for Medical Research, K. U. Leuven, Minderbroedersstraat 10, B-3000 Leuven, Belgium.
  • Menéndez-Arias L; Centro de Biología Molecular "Severo Ochoa" (Consejo Superior de Investigaciones Científicas & Universidad Autónoma de Madrid), Madrid, Spain. Electronic address: lmenendez@cbm.csic.es.
  • Zhan P; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China. Electronic address: zhanpeng1982@sdu.edu.cn.
  • Liu X; Department of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Ji'nan 250012, PR China. Electronic address: xinyongl@sdu.edu.cn.
Bioorg Med Chem ; 30: 115927, 2021 01 15.
Article en En | MEDLINE | ID: mdl-33352387
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Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Sulfonas / VIH-1 / Inhibidores de la Transcriptasa Inversa / Fármacos Anti-VIH / Transcriptasa Inversa del VIH / Indoles Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2021 Tipo del documento: Article
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Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Sulfonas / VIH-1 / Inhibidores de la Transcriptasa Inversa / Fármacos Anti-VIH / Transcriptasa Inversa del VIH / Indoles Idioma: En Revista: Bioorg Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2021 Tipo del documento: Article