In vitro and in vivo assessment of hydroxypropyl cellulose as functional additive for enabling formulations containing itraconazole.
Int J Pharm X
; 3: 100076, 2021 Dec.
Article
en En
| MEDLINE
| ID: mdl-33851133
API, active pharmaceutical ingredient; ASD, amorphous solid dispersion; AUC, area under the curve; AcN, acetonitrile; Amorphous solid dispersion; BCS, biopharmaceutical classification system; Biphasic dissolution; DMSO, dimethyl sulfoxide; DSC, differential scanning calorimetry; FaSSIF, fasted state simulated intestinal fluid; GI, gastrointestinal; HME, hot-melt extrusion; HPC; HPC, hydroxypropyl cellulose; HPMC; HPMC, hydroxypropyl methyl cellulose; Hot-melt extrusion; ITZ, itraconazole; KTZ, ketoconazole; NCE, new chemical entity; OH-ITZ, hydroxy-itraconazole; PM, physical mixture; SD, spray-drying; TG, glass transition temperature; XRPD, x-ray powder diffraction
Texto completo:
1
Bases de datos:
MEDLINE
Tipo de estudio:
Prognostic_studies
Idioma:
En
Revista:
Int J Pharm X
Año:
2021
Tipo del documento:
Article
País de afiliación:
Alemania