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Discovery of a Potent and Selective Covalent p300/CBP Inhibitor.
Mastracchio, Anthony; Lai, Chunqiu; Digiammarino, Enrico; Ready, Damien B; Lasko, Loren M; Bromberg, Kenneth D; McClellan, William J; Montgomery, Debra; Manaves, Vlasios; Shaw, Bailin; Algire, Mikkel; Patterson, Melanie J; Sun, Chaohong C; Rosenberg, Saul; Lai, Albert; Michaelides, Michael R.
Afiliación
  • Mastracchio A; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Lai C; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Digiammarino E; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Ready DB; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Lasko LM; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Bromberg KD; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • McClellan WJ; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Montgomery D; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Manaves V; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Shaw B; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Algire M; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Patterson MJ; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Sun CC; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Rosenberg S; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Lai A; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
  • Michaelides MR; AbbVie, Inc., 1 North Waukegan Road, North Chicago, Illinois 60064, United States.
ACS Med Chem Lett ; 12(5): 726-731, 2021 May 13.
Article en En | MEDLINE | ID: mdl-34055218

Texto completo: 1 Bases de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Bases de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2021 Tipo del documento: Article País de afiliación: Estados Unidos