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Metabolism, pharmacokinetics, and anticonvulsant activity of a deuterated analog of the α2/3-selective GABAkine KRM-II-81.
Golani, Lalit K; Divovic, Branka; Sharmin, Dishary; Pandey, Kamal P; Mian, Md Yeunus; Cerne, Rok; Zahn, Nicolas M; Meyer, Michelle J; Tiruveedhula, Veera V N P B; Smith, Jodi L; Ping, Xingjie; Jin, Xiaoming; Lippa, Arnold; Schkeryantz, Jeffrey M; Arnold, Leggy A; Cook, James M; Savic, Miroslav M; Witkin, Jeffrey M.
Afiliación
  • Golani LK; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
  • Divovic B; Department of Pharmacology, Faculty of Pharmacy, University of Belgrade, Belgrade, Serbia.
  • Sharmin D; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
  • Pandey KP; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
  • Mian MY; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
  • Cerne R; Laboratory of Antiepileptic Drug Discovery, Ascencion St. Vincent, Indianapolis, Indiana, USA.
  • Zahn NM; Department of Anatomy and Cell Biology, Indiana University/Purdue University, Indianapolis, Indiana, USA.
  • Meyer MJ; Faculty of Medicine, University of Ljubljana, Ljubljana, Slovenia.
  • Tiruveedhula VVNPB; RespireRx Pharmaceuticals Inc, Glen Rock, New Jersey, USA.
  • Smith JL; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
  • Ping X; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
  • Jin X; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
  • Lippa A; Laboratory of Antiepileptic Drug Discovery, Ascencion St. Vincent, Indianapolis, Indiana, USA.
  • Schkeryantz JM; Department of Anatomy and Cell Biology, Indiana University/Purdue University, Indianapolis, Indiana, USA.
  • Arnold LA; Department of Anatomy and Cell Biology, Indiana University/Purdue University, Indianapolis, Indiana, USA.
  • Cook JM; RespireRx Pharmaceuticals Inc, Glen Rock, New Jersey, USA.
  • Savic MM; Bristol Myers Squibb, Cambridge, Massachusetts, USA.
  • Witkin JM; Department of Chemistry & Biochemistry, Milwaukee Institute of Drug Discovery, University of Wisconsin-Milwaukee, Milwaukee, Wisconsin, USA.
Biopharm Drug Dispos ; 43(2): 66-75, 2022 Apr.
Article en En | MEDLINE | ID: mdl-35194800

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Antibióticos Antituberculosos / Anticonvulsivantes Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Revista: Biopharm Drug Dispos Año: 2022 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Antibióticos Antituberculosos / Anticonvulsivantes Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Revista: Biopharm Drug Dispos Año: 2022 Tipo del documento: Article País de afiliación: Estados Unidos