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A novel small-molecule selective activator of homomeric GIRK4 channels.
Cui, Meng; Xu, Keman; Gada, Kirin D; Shalomov, Boris; Ban, Michelle; Eptaminitaki, Giasemi C; Kawano, Takeharu; Plant, Leigh D; Dascal, Nathan; Logothetis, Diomedes E.
Afiliación
  • Cui M; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA; Center for Drug Discovery, Northeastern University, Boston, Massachusetts, USA. Electronic address: m.cui@northeastern.edu.
  • Xu K; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA.
  • Gada KD; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA.
  • Shalomov B; Department of Physiology and Pharmacology and Sagol School of Neuroscience, School of Medicine, Tel Aviv University, Tel Aviv, Israel.
  • Ban M; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA.
  • Eptaminitaki GC; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA.
  • Kawano T; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA.
  • Plant LD; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA; Center for Drug Discovery, Northeastern University, Boston, Massachusetts, USA.
  • Dascal N; Department of Physiology and Pharmacology and Sagol School of Neuroscience, School of Medicine, Tel Aviv University, Tel Aviv, Israel.
  • Logothetis DE; Department of Pharmaceutical Sciences, School of Pharmacy, Bouvé College of Health Sciences, Northeastern University, Boston, Massachusetts, USA; Center for Drug Discovery, Northeastern University, Boston, Massachusetts, USA; Chemistry and Chemical Biology, College of Science, Northeastern Universit
J Biol Chem ; 298(6): 102009, 2022 06.
Article en En | MEDLINE | ID: mdl-35525275

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Canales de Potasio Rectificados Internamente Asociados a la Proteína G / Indoles Límite: Humans Idioma: En Revista: J Biol Chem Año: 2022 Tipo del documento: Article

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Canales de Potasio Rectificados Internamente Asociados a la Proteína G / Indoles Límite: Humans Idioma: En Revista: J Biol Chem Año: 2022 Tipo del documento: Article