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Discovery of a new class of triazole based inhibitors of acetyl transferase KAT2A.
Pacifico, Roberta; Del Gaudio, Nunzio; Bove, Guglielmo; Altucci, Lucia; Siragusa, Lydia; Cruciani, Gabriele; Ruvo, Menotti; Bellavita, Rosa; Grieco, Paolo; Adamo, Mauro F A.
Afiliación
  • Pacifico R; Centre for Synthesis and Chemical Biology (CSCB), Department of Chemistry, Royal College of Surgeons in Ireland, Dublin, Ireland.
  • Del Gaudio N; Department of precision medicine, University of Campania Luigi Vanvitelli, Naples, Italy.
  • Bove G; Department of precision medicine, University of Campania Luigi Vanvitelli, Naples, Italy.
  • Altucci L; Department of precision medicine, University of Campania Luigi Vanvitelli, Naples, Italy.
  • Siragusa L; Molecular Horizon Srl, Bettona, Italy.
  • Cruciani G; Laboratory for Chemometrics and Molecular Modeling, Department of Chemistry, Biology, and Biotechnology, University of Perugia, Perugia, Italy.
  • Ruvo M; Institute of Biostructures and Bioimaging, Consiglio Nazionale delle Ricerche, Naples, Italy.
  • Bellavita R; Department of Pharmacy, School of Medicine, University of Naples 'Federico II', Naples, Italy.
  • Grieco P; Department of Pharmacy, School of Medicine, University of Naples 'Federico II', Naples, Italy.
  • Adamo MFA; Centre for Synthesis and Chemical Biology (CSCB), Department of Chemistry, Royal College of Surgeons in Ireland, Dublin, Ireland.
J Enzyme Inhib Med Chem ; 37(1): 1987-1994, 2022 Dec.
Article en En | MEDLINE | ID: mdl-35880250

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Acetiltransferasas / Triazoles Tipo de estudio: Prognostic_studies Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Irlanda

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Acetiltransferasas / Triazoles Tipo de estudio: Prognostic_studies Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2022 Tipo del documento: Article País de afiliación: Irlanda