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Optimization of pyridylpiperazine-based inhibitors of the Escherichia coli AcrAB-TolC efflux pump.
Compagne, Nina; Jiménez-Castellanos, Juan-Carlos; Meurillon, Virginie; Pradel, Elizabeth; Vieira Da Cruz, Anais; Piveteau, Catherine; Biela, Alexandre; Eveque, Maxime; Leroux, Florence; Deprez, Benoit; Willand, Nicolas; Hartkoorn, Ruben C; Flipo, Marion.
Afiliación
  • Compagne N; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Jiménez-Castellanos JC; Univ. Lille, CNRS, Inserm, CHU Lille, Institut Pasteur de Lille, U1019 - UMR 9017 - CIIL - Center for Infection and Immunity of Lille, F-59000, Lille, France.
  • Meurillon V; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Pradel E; Univ. Lille, CNRS, Inserm, CHU Lille, Institut Pasteur de Lille, U1019 - UMR 9017 - CIIL - Center for Infection and Immunity of Lille, F-59000, Lille, France.
  • Vieira Da Cruz A; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Piveteau C; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Biela A; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Eveque M; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Leroux F; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France; Univ. Lille, CNRS, Inserm, CHU Lille, Institut Pasteur Lille, US 41-UAR 2014-PLBS, F-59000, Lille, France.
  • Deprez B; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Willand N; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France.
  • Hartkoorn RC; Univ. Lille, CNRS, Inserm, CHU Lille, Institut Pasteur de Lille, U1019 - UMR 9017 - CIIL - Center for Infection and Immunity of Lille, F-59000, Lille, France. Electronic address: ruben.hartkoorn@inserm.fr.
  • Flipo M; Univ. Lille, Inserm, Institut Pasteur de Lille, U1177-Drugs and Molecules for Living Systems, F-59000, Lille, France. Electronic address: marion.flipo@univ-lille.fr.
Eur J Med Chem ; 259: 115630, 2023 Nov 05.
Article en En | MEDLINE | ID: mdl-37459793

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Proteínas de Escherichia coli / Escherichia coli Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: Francia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Proteínas de Escherichia coli / Escherichia coli Idioma: En Revista: Eur J Med Chem Año: 2023 Tipo del documento: Article País de afiliación: Francia