1.
Beilstein J Org Chem
; 14: 1452-1458, 2018.
Artigo
em Inglês
| MEDLINE
| ID: mdl-29977409
RESUMO
The reaction of enamine compounds with the Togni reagent in the presence of CuI afforded ß-trifluoromethylated enamine intermediates, which were converted directly to biologically interesting trifluoromethylated 2H-azirines by an iodosobenzene (PhIO)-mediated intramolecular azirination in a one-pot process.