Detalhe da pesquisa
1.
Serendipitous Identification of a Covalent Activator of Liver Pyruvate Kinase.
Chembiochem
; 24(1): e202200339, 2023 01 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-36250581
2.
Synthesis and in vivo evaluation of [11C]tucatinib for HER2-targeted PET imaging.
Bioorg Med Chem Lett
; 80: 129088, 2023 01 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-36455802
3.
Synthesis and radiolabeling of a polar [125 I]I-1,2,4,5-tetrazine.
J Labelled Comp Radiopharm
; 66(1): 22-30, 2023 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-36539610
4.
Development of the First Tritiated Tetrazine: Facilitating Tritiation of Proteins.
Chembiochem
; 23(23): e202200539, 2022 12 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-36333105
5.
[11 C]Carboxylated Tetrazines for Facile Labeling of Trans-Cyclooctene-Functionalized PeptoBrushes.
Macromol Rapid Commun
; 43(12): e2100655, 2022 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-34888977
6.
Optimization of Direct Aromatic 18F-Labeling of Tetrazines.
Molecules
; 27(13)2022 Jun 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-35807267
7.
A Metabolomic Approach Applied to a Liquid Chromatography Coupled to High-Resolution Tandem Mass Spectrometry Method (HPLC-ESI-HRMS/MS): Towards the Comprehensive Evaluation of the Chemical Composition of Cannabis Medicinal Extracts.
Phytochem Anal
; 29(2): 144-155, 2018 Mar.
Artigo
em Inglês
| MEDLINE | ID: mdl-28915313
8.
Design, stereoselective synthesis, configurational stability and biological activity of 7-chloro-9-(furan-3-yl)-2,3,3a,4-tetrahydro-1H-benzo[e]pyrrolo[2,1-c][1,2,4]thiadiazine 5,5-dioxide.
Bioorg Med Chem
; 22(17): 4667-76, 2014 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-25126714
9.
Sulfone-based human liver pyruvate kinase inhibitors - Design, synthesis and in vitro bioactivity.
Eur J Med Chem
; 269: 116306, 2024 Apr 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-38471358
10.
Exploration of Novel Urolithin C Derivatives as Non-Competitive Inhibitors of Liver Pyruvate Kinase.
Pharmaceuticals (Basel)
; 16(5)2023 Apr 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-37242451
11.
Next generation fibroblast activation protein (FAP) targeting PET tracers - The tetrazine ligation allows an easy and convenient way to 18F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines.
Eur J Med Chem
; 262: 115862, 2023 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37883899
12.
Ellagic Acid and Its Metabolites as Potent and Selective Allosteric Inhibitors of Liver Pyruvate Kinase.
Nutrients
; 15(3)2023 Jan 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-36771285
13.
Pretargeted imaging beyond the blood-brain barrier.
RSC Med Chem
; 14(3): 444-453, 2023 Mar 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-36970152
14.
Recent Advances in the Development of Tetrazine Ligation Tools for Pretargeted Nuclear Imaging.
Pharmaceuticals (Basel)
; 15(6)2022 May 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-35745604
15.
Development of 18F-Labeled Bispyridyl Tetrazines for In Vivo Pretargeted PET Imaging.
Pharmaceuticals (Basel)
; 15(2)2022 Feb 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-35215356
16.
Evaluation of the α-synuclein PET radiotracer (d3)-[11C]MODAG-001 in pigs.
Nucl Med Biol
; 114-115: 42-48, 2022.
Artigo
em Inglês
| MEDLINE | ID: mdl-36095921
17.
Insights into Elution of Anion Exchange Cartridges: Opening the Path toward Aliphatic 18F-Radiolabeling of Base-Sensitive Tracers.
ACS Pharmacol Transl Sci
; 4(5): 1556-1566, 2021 Oct 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-34661074
18.
Alpha-Synuclein PET Tracer Development-An Overview about Current Efforts.
Pharmaceuticals (Basel)
; 14(9)2021 Aug 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-34577548
19.
Synthesis and biological evaluation of 1,3-dioxolane-based 5-HT1A receptor agonists for CNS disorders and neuropathic pain.
Future Med Chem
; 10(18): 2137-2154, 2018 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-30043643
20.
Structure-Activity Relationships within a Series of σ1 and σ2 Receptor Ligands: Identification of a σ2 Receptor Agonist (BS148) with Selective Toxicity against Metastatic Melanoma.
ChemMedChem
; 12(22): 1893-1905, 2017 11 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-28940806