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Bioorg Med Chem Lett
; 14(13): 3441-4, 2004 Jul 05.
Artigo
em Inglês
| MEDLINE
| ID: mdl-15177449
RESUMO
2,5-Dihydropyrazolo[4,3-c]pyridin-3-ones are GABAA receptor benzodiazepine binding site ligands with functional selectivity for the alpha3 subtype over the alpha1 subtype. SAR studies to optimise this functional selectivity are described.