Detalhe da pesquisa
1.
Synthesis and Pharmacological Evaluation of Enantiopure N-Substituted Ortho-c Oxide-Bridged 5-Phenylmorphans.
Molecules
; 27(24)2022 Dec 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-36557961
2.
Design, Synthesis, and In Vivo Evaluation of C1-Linked 4,5-Epoxymorphinan Haptens for Heroin Vaccines.
Molecules
; 27(5)2022 Feb 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-35268659
3.
X-ray Crystallography and Unexpected Chiroptical Properties Reassign the Configuration of Haliclonadiamine.
J Am Chem Soc
; 142(6): 2755-2759, 2020 02 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-31986017
4.
Reaction Kinetics Direct a Rational Synthesis of an HIV-1 Inactivator of Nucleocapsid Protein 7 and Provide Mechanistic Insight into Cellular Metabolism and Antiviral Activity.
Chemistry
; 24(38): 9485-9489, 2018 Jul 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-29653024
5.
Total Synthesis of Sarpagine-Related Bioactive Indole Alkaloids.
Chemistry
; 24(10): 2354-2359, 2018 Feb 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-29244896
6.
A High Aspect Ratio Bifurcated 128-Microchannel Microfluidic Device for Environmental Monitoring of Explosives.
Sensors (Basel)
; 18(5)2018 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-29762499
7.
Engineering Immunological Tolerance Using Quantum Dots to Tune the Density of Self-Antigen Display.
Adv Funct Mater
; 27(22)2017 Jun 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-29503604
8.
Concise Total Synthesis of (-)-Affinisine Oxindole, (+)-Isoalstonisine, (+)-Alstofoline, (-)-Macrogentine, (+)-Na -Demethylalstonisine, (-)-Alstonoxineâ A, and (+)-Alstonisine.
Chemistry
; 23(62): 15805-15819, 2017 Nov 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-28875520
9.
Iodobenzene-Catalyzed Synthesis of Phenanthridinones via Oxidative C-H Amidation.
J Org Chem
; 82(7): 3589-3596, 2017 04 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-28245353
10.
One-pot sequential reaction to 2-substituted-phenanthridinones from N-methoxybenzamides.
Org Biomol Chem
; 15(20): 4390-4398, 2017 May 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-28475192
11.
Modulation of opioid receptor affinity and efficacy via N-substitution of 9ß-hydroxy-5-(3-hydroxyphenyl)morphan: Synthesis and computer simulation study.
Bioorg Med Chem
; 25(8): 2406-2422, 2017 04 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-28314512
12.
Design, Synthesis, and Biological Evaluation of Structurally Rigid Analogues of 4-(3-Hydroxyphenyl)piperidine Opioid Receptor Antagonists.
J Org Chem
; 81(21): 10383-10391, 2016 11 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-27462910
13.
Efficacy, but not antibody titer or affinity, of a heroin hapten conjugate vaccine correlates with increasing hapten densities on tetanus toxoid, but not on CRM197 carriers.
Bioconjug Chem
; 26(6): 1041-53, 2015 Jun 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-25970207
14.
Synthesis of aza and carbocyclic ß-carbolines for the treatment of alcohol abuse. Regiospecific solution to the problem of 3,6-disubstituted ß- and aza-ß-carboline specificity.
Org Biomol Chem
; 13(43): 10705-15, 2015 Nov 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-26349488
15.
PABA/NO lead optimization: Improved targeting of cytotoxicity to glutathione S-transferase P1-overexpressing cancer cells.
Bioorg Med Chem
; 23(15): 4980-4988, 2015 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26043946
16.
Using click chemistry toward novel 1,2,3-triazole-linked dopamine D3 receptor ligands.
Bioorg Med Chem
; 23(14): 4000-12, 2015 Jul 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-25650314
17.
Chiral resolution and absolute configuration of the enantiomers of the psychoactive "designer drug" 3,4-methylenedioxypyrovalerone.
Chirality
; 27(4): 287-93, 2015 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-25727807
18.
Synthesis of 1,2-dihydro-2-oxo-4-quinolinyl phosphates from 2-acyl-benzoic acids.
Tetrahedron Lett
; 56(11): 1441-1444, 2015 Mar 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-25937677
19.
General strategy for synthesis of C-19 methyl-substituted sarpagine/macroline/ajmaline indole alkaloids including total synthesis of 19(S),20(R)-dihydroperaksine, 19(S),20(R)-dihydroperaksine-17-al, and peraksine.
J Org Chem
; 79(21): 10030-48, 2014 Nov 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-25247616
20.
Synthesis of enantiopure 10-nornaltrexones in the search for Toll-like receptor 4 antagonists and opioid ligands.
J Org Chem
; 79(11): 5007-18, 2014 Jun 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-24773391