Detalhe da pesquisa
1.
An Efficient Way to Screen Inhibitors of Energy-Coupling Factor (ECF) Transporters in a Bacterial Uptake Assay.
Int J Mol Sci
; 23(5)2022 Feb 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-35269783
2.
Harnessing the 12 Green Chemistry Principles for Sustainable Antiparasitic Drugs: Toward the One Health Approach.
ACS Infect Dis
; 2024 May 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-38724015
3.
Hit optimization by dynamic combinatorial chemistry on Streptococcus pneumoniae energy-coupling factor transporter ECF-PanT.
Chem Commun (Camb)
; 60(7): 870-873, 2024 Jan 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-38164786
4.
Click Chemistry and Targeted Degradation: A Winning Combination for Medicinal Chemists?
ChemMedChem
; 18(20): e202300422, 2023 10 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-37706617
5.
Back in Person: Frontiers in Medicinal Chemistry 2023.
ChemMedChem
; 18(19): e202300344, 2023 10 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-37485831
6.
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors.
ChemMedChem
; 18(19): e202300346, 2023 10 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-37718320
7.
Identification of inhibitors targeting the energy-coupling factor (ECF) transporters.
Commun Biol
; 6(1): 1182, 2023 11 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-37985798
8.
Favourable involvement of α2A-adrenoreceptor antagonism in the I2-imidazoline binding sites-mediated morphine analgesia enhancement.
Bioorg Med Chem
; 20(7): 2259-65, 2012 Apr 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-22370341
9.
Might the observed α(2A)-adrenoreceptor agonism or antagonism of allyphenyline analogues be ascribed to different molecular conformations?
Bioorg Med Chem
; 20(6): 2082-90, 2012 Mar 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-22341244
10.
Structure-Guided Optimization of Small-Molecule Folate Uptake Inhibitors Targeting the Energy-Coupling Factor Transporters.
J Med Chem
; 65(13): 8869-8880, 2022 07 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-35709475
11.
Frontiers in Medicinal Chemistry 2022 Goes Virtual.
ChemMedChem
; 17(21): e202200419, 2022 Nov 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-36198574
12.
Targeting the IspD Enzyme in the MEP Pathway: Identification of a Novel Fragment Class.
ChemMedChem
; 17(5): e202100679, 2022 03 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-34918860
13.
Bacteriomimetic Liposomes Improve Antibiotic Activity of a Novel Energy-Coupling Factor Transporter Inhibitor.
Pharmaceutics
; 14(1)2021 Dec 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-35056900
14.
Assessment of the rules related to gaining activity against Gram-negative bacteria.
RSC Med Chem
; 12(4): 593-601, 2021 Apr 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-34046630
15.
Search for the Active Ingredients from a 2-Aminothiazole DMSO Stock Solution with Antimalarial Activity.
ChemMedChem
; 16(13): 2089-2093, 2021 07 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-33844432
16.
Author Correction: Identification of inhibitors targeting the energy-coupling factor (ECF) transporters.
Commun Biol
; 7(1): 70, 2024 Jan 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-38195913
17.
CD1b Tetramers Identify T Cells that Recognize Natural and Synthetic Diacylated Sulfoglycolipids from Mycobacterium tuberculosis.
Cell Chem Biol
; 25(4): 392-402.e14, 2018 04 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-29398561
18.
DXS as a target for structure-based drug design.
Future Med Chem
; 9(11): 1277-1294, 2017 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-28636418
19.
Synthesis and characterization of the first inhibitor of N-acylphosphatidylethanolamine phospholipase D (NAPE-PLD).
Chem Commun (Camb)
; 53(95): 12814-12817, 2017 Nov 28.
Artigo
em Inglês
| MEDLINE | ID: mdl-29143042
20.
Combined Interactions with I1-, I2-Imidazoline Binding Sites and α2-Adrenoceptors To Manage Opioid Addiction.
ACS Med Chem Lett
; 7(10): 956-961, 2016 Oct 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-27774136