Detalhe da pesquisa
1.
Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity.
bioRxiv
; 2024 Feb 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-38405908
2.
Structural Basis for Highly Selective Class II Alpha Phosphoinositide-3-Kinase Inhibition.
J Med Chem
; 66(20): 14278-14302, 2023 10 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-37819647