Detalhe da pesquisa
1.
Identification of a series of 4-[3-(quinolin-2-yl)-1,2,4-oxadiazol-5-yl]piperazinyl ureas as potent smoothened antagonist hedgehog pathway inhibitors.
Bioorg Med Chem Lett
; 21(18): 5274-82, 2011 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21803580
2.
Identification of substituted pyrazolo[1,5-a]quinazolin-5(4H)-one as potent poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors.
Bioorg Med Chem Lett
; 19(15): 4196-200, 2009 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-19541484
3.
2-(2-Thienyl)-5,6-dihydroxy-4-carboxypyrimidines as inhibitors of the hepatitis C virus NS5B polymerase: discovery, SAR, modeling, and mutagenesis.
J Med Chem
; 49(5): 1693-705, 2006 Mar 09.
Artigo
em Inglês
| MEDLINE | ID: mdl-16509585
4.
Discovery of 2-{4-[(3S)-piperidin-3-yl]phenyl}-2H-indazole-7-carboxamide (MK-4827): a novel oral poly(ADP-ribose)polymerase (PARP) inhibitor efficacious in BRCA-1 and -2 mutant tumors.
J Med Chem
; 52(22): 7170-85, 2009 Nov 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-19873981