Detalhe da pesquisa
1.
The decanoate esters of nandrolone, testosterone, and trenbolone induce steroid specific memory impairment and somatic effects in the male rat.
Horm Behav
; 161: 105501, 2024 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-38368844
2.
The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds.
Int J Mol Sci
; 25(7)2024 Apr 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-38612894
3.
Inhibition of Insulin-Regulated Aminopeptidase by Imidazo [1,5-α]pyridines-Synthesis and Evaluation.
Int J Mol Sci
; 25(5)2024 Feb 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-38473764
4.
Two-Chamber Aminocarbonylation of Aryl Bromides and Triflates Using Amino Acids as Nucleophiles.
J Org Chem
; 88(18): 12978-12985, 2023 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37639573
5.
Hydrogen Peroxide Induced Toxicity Is Reversed by the Macrocyclic IRAP-Inhibitor HA08 in Primary Hippocampal Cell Cultures.
Curr Issues Mol Biol
; 44(10): 5000-5012, 2022 Oct 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-36286055
6.
2-Alkyl substituted benzimidazoles as a new class of selective AT2 receptor ligands.
Bioorg Med Chem
; 66: 116804, 2022 07 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-35576659
7.
N-(Methyloxycarbonyl)thiophene sulfonamides as high affinity AT2 receptor ligands.
Bioorg Med Chem
; 29: 115859, 2021 01 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-33309749
8.
Design, synthesis and in vitro biological evaluation of oligopeptides targeting E. coli type I signal peptidase (LepB).
Bioorg Med Chem
; 25(3): 897-911, 2017 02 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-28038943
9.
Discovery of pyrazinone based compounds that potently inhibit the drug-resistant enzyme variant R155K of the hepatitis C virus NS3 protease.
Bioorg Med Chem
; 24(12): 2603-20, 2016 06 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-27160057
10.
Toward Biomass-Based Organic Electronics: Continuous Flow Synthesis and Electropolymerization of N-Substituted Pyrroles.
ACS Omega
; 9(12): 13852-13859, 2024 Mar 26.
Artigo
em Inglês
| MEDLINE | ID: mdl-38559979
11.
N-(Heteroaryl)thiophene sulfonamides as angiotensin AT2 receptor ligands.
Eur J Med Chem
; 265: 116122, 2024 Feb 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-38199164
12.
Microwave-assisted synthesis of small molecules targeting the infectious diseases tuberculosis, HIV/AIDS, malaria and hepatitis C.
Org Biomol Chem
; 10(14): 2713-29, 2012 Apr 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-22227602
13.
Diastereoselective Synthesis of N-Methylspiroindolines by Intramolecular Mizoroki-Heck Annulations.
ACS Omega
; 7(36): 32525-32535, 2022 Sep 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-36120037
14.
Discovery of achiral inhibitors of the hepatitis C virus NS3 protease based on 2(1H)-pyrazinones.
Bioorg Med Chem
; 18(17): 6512-25, 2010 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-20673728
15.
Functionalized 3-amino-imidazo[1,2-a]pyridines: a novel class of drug-like Mycobacterium tuberculosis glutamine synthetase inhibitors.
Bioorg Med Chem Lett
; 19(16): 4790-3, 2009 Aug 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-19560924
16.
A straightforward microwave method for rapid synthesis of N-1, C-6 functionalized 3,5-dichloro-2(1H)-pyrazinones.
Org Biomol Chem
; 7(13): 2809-15, 2009 Jul 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-19532999
17.
A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode.
ChemistryOpen
; 8(1): 114-125, 2019 Jan.
Artigo
em Inglês
| MEDLINE | ID: mdl-30697513
18.
ENABLE: an engine for European antibacterial drug discovery and development.
Nat Rev Drug Discov
; 20(6): 407-408, 2021 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-33948003
19.
Optimization and Evaluation of 5-Styryl-Oxathiazol-2-one Mycobacterium tuberculosis Proteasome Inhibitors as Potential Antitubercular Agents.
ChemistryOpen
; 4(3): 342-62, 2015 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-26246997
20.
Syntheses of new tuberculosis inhibitors promoted by microwave irradiation.
Ups J Med Sci
; 119(2): 181-91, 2014 May.
Artigo
em Inglês
| MEDLINE | ID: mdl-24666224