Detalhe da pesquisa
1.
Rapid Construction of a Chloromethyl-Substituted Duocarmycin-like Prodrug.
Molecules
; 28(12)2023 Jun 16.
Artigo
em Inglês
| MEDLINE | ID: mdl-37375372
2.
Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses.
J Am Chem Soc
; 144(7): 2905-2920, 2022 02 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-35142215
3.
Discovery of novel pyrrolopyridazine scaffolds as transient receptor potential vanilloid (TRPV1) antagonists.
Bioorg Med Chem Lett
; 22(22): 6888-95, 2012 Nov 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-23058884
4.
Phenyl isoxazole voltage-gated sodium channel blockers: structure and activity relationship.
Bioorg Med Chem Lett
; 21(13): 3871-6, 2011 Jul 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21641215
5.
The Oncolytic Efficacy and in Vivo Pharmacokinetics of [2-(4-Chlorophenyl)quinolin-4-yl](piperidine-2-yl)methanol (Vacquinol-1) Are Governed by Distinct Stereochemical Features.
J Med Chem
; 59(18): 8577-92, 2016 09 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-27607569
6.
Creation of Novel Cores for ß-Secretase (BACE-1) Inhibitors: A Multiparameter Lead Generation Strategy.
ACS Med Chem Lett
; 5(4): 440-5, 2014 Apr 10.
Artigo
em Inglês
| MEDLINE | ID: mdl-24900855
7.
Core refinement toward permeable ß-secretase (BACE-1) inhibitors with low hERG activity.
J Med Chem
; 56(11): 4181-205, 2013 Jun 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-23126626
8.
New aminoimidazoles as ß-secretase (BACE-1) inhibitors showing amyloid-ß (Aß) lowering in brain.
J Med Chem
; 55(21): 9297-311, 2012 Nov 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-23017051