Detalhe da pesquisa
1.
The Impact of Nε-Acryloyllysine Piperazides on the Conformational Dynamics of Transglutaminase 2.
Int J Mol Sci
; 24(2)2023 Jan 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-36675164
2.
Fluorescence Anisotropy Assay with Guanine Nucleotides Provides Access to Functional Analysis of Gαi1 Proteins.
Anal Chem
; 94(41): 14410-14418, 2022 10 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-36206384
3.
Application of a Fluorescence Anisotropy-Based Assay to Quantify Transglutaminase 2 Activity in Cell Lysates.
Int J Mol Sci
; 23(9)2022 Apr 19.
Artigo
em Inglês
| MEDLINE | ID: mdl-35562866
4.
Solid-Phase Synthesis of Selectively Mono-Fluorobenz(o)ylated Polyamines as a Basis for the Development of 18F-Labeled Radiotracers.
Molecules
; 26(22)2021 Nov 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-34834103
5.
Solution-phase synthesis of the fluorogenic TGase 2 acyl donor Z-Glu(HMC)-Gly-OH and its use for inhibitor and amine substrate characterisation.
Anal Biochem
; 595: 113612, 2020 04 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32045569
6.
The Pyrazolo[3,4-d]pyrimidine-Based Kinase Inhibitor NVP-BHG712: Effects of Regioisomers on Tumor Growth, Perfusion, and Hypoxia in EphB4-Positive A375 Melanoma Xenografts.
Molecules
; 25(21)2020 Nov 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-33153234
7.
Synthesis, 18F-labelling and radiopharmacological characterisation of the C-terminal 30mer of Clostridium perfringens enterotoxin as a potential claudin-targeting peptide.
Amino Acids
; 51(2): 219-244, 2019 Feb.
Artigo
em Inglês
| MEDLINE | ID: mdl-30264172
8.
Cathepsin B: Active site mapping with peptidic substrates and inhibitors.
Bioorg Med Chem
; 27(1): 1-15, 2019 01 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-30473362
9.
Synthesis and preliminary radiopharmacological characterisation of an 11 C-labelled azadipeptide nitrile as potential PET tracer for imaging of cysteine cathepsins.
J Labelled Comp Radiopharm
; 62(8): 448-459, 2019 06 30.
Artigo
em Inglês
| MEDLINE | ID: mdl-30912586
10.
A fluorescence anisotropy-based assay for determining the activity of tissue transglutaminase.
Amino Acids
; 49(3): 567-583, 2017 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-26886924
11.
Synthesis and Kinetic Characterisation of Water-Soluble Fluorogenic Acyl Donors for Transglutaminaseâ 2.
Chembiochem
; 17(13): 1263-81, 2016 07 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27124709
12.
Targeting lysyl oxidase for molecular imaging in breast cancer.
Breast Cancer Res
; 17: 107, 2015 Aug 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-26265048
13.
Cyclopeptides containing the DEKS motif as conformationally restricted collagen telopeptide analogues: synthesis and conformational analysis.
Org Biomol Chem
; 13(6): 1878-96, 2015 Feb 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-25503999
14.
Preclinical evaluation of an 18F-labeled Nε-acryloyllysine piperazide for covalent targeting of transglutaminase 2.
EJNMMI Radiopharm Chem
; 9(1): 1, 2024 Jan 02.
Artigo
em Inglês
| MEDLINE | ID: mdl-38165538
15.
Tissue transglutaminase: an emerging target for therapy and imaging.
Bioorg Med Chem Lett
; 23(24): 6528-43, 2013 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-24432384
16.
Use of 3-[(18)F]fluoropropanesulfonyl chloride as a prosthetic agent for the radiolabelling of amines: Investigation of precursor molecules, labelling conditions and enzymatic stability of the corresponding sulfonamides.
Beilstein J Org Chem
; 9: 1002-11, 2013.
Artigo
em Inglês
| MEDLINE | ID: mdl-23766817
17.
Comparative Saturation Binding Analysis of 64Cu-Labeled Somatostatin Analogues Using Cell Homogenates and Intact Cells.
ACS Omega
; 8(26): 24003-24009, 2023 Jul 04.
Artigo
em Inglês
| MEDLINE | ID: mdl-37426243
18.
Lysyl Oxidases as Targets for Cancer Therapy and Diagnostic Imaging.
ChemMedChem
; 18(18): e202300331, 2023 09 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37565736
19.
Enzymological Characterization of 64Cu-Labeled Neprilysin Substrates and Their Application for Modulating the Renal Clearance of Targeted Radiopharmaceuticals.
J Med Chem
; 66(1): 516-537, 2023 01 12.
Artigo
em Inglês
| MEDLINE | ID: mdl-36595224
20.
Dipeptide-Derived Alkynes as Potent and Selective Irreversible Inhibitors of Cysteine Cathepsins.
J Med Chem
; 66(6): 3818-3851, 2023 03 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-36867428