Detalhe da pesquisa
1.
Crossing of the Cystic Barriers of Toxoplasma gondii by the Fluorescent Coumarin Tetra-Cyclopeptide.
Molecules
; 26(24)2021 Dec 11.
Artigo
em Inglês
| MEDLINE | ID: mdl-34946588
2.
Inhibitors of ABCG2-mediated multidrug resistance: Lead generation through computer-aided drug design.
Eur J Med Chem
; 248: 115070, 2023 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-36628850
3.
Resorcinol-based hemiindigoid derivatives as human tyrosinase inhibitors and melanogenesis suppressors in human melanoma cells.
Eur J Med Chem
; 246: 114972, 2023 Jan 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-36462443
4.
Characterization of Potent ABCG2 Inhibitor Derived from Chromone: From the Mechanism of Inhibition to Human Extracellular Vesicles for Drug Delivery.
Pharmaceutics
; 15(4)2023 Apr 17.
Artigo
em Inglês
| MEDLINE | ID: mdl-37111745
5.
Design, synthesis and pharmacological evaluation of novel naphthalenic derivatives as selective MT(1) melatoninergic ligands.
Bioorg Med Chem
; 18(10): 3426-36, 2010 May 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-20444610
6.
Advances in the Design of Genuine Human Tyrosinase Inhibitors for Targeting Melanogenesis and Related Pigmentations.
J Med Chem
; 63(22): 13428-13443, 2020 11 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-32787103
7.
Chromones bearing amino acid residues: Easily accessible and potent inhibitors of the breast cancer resistance protein ABCG2.
Eur J Med Chem
; 202: 112503, 2020 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32653696
8.
Molecular analysis of the massive GSH transport mechanism mediated by the human Multidrug Resistant Protein 1/ABCC1.
Sci Rep
; 10(1): 7616, 2020 05 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-32377003
9.
Optimization of the chromone scaffold through QSAR and docking studies: Identification of potent inhibitors of ABCG2.
Eur J Med Chem
; 184: 111772, 2019 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-31630055
10.
Aurone derivatives as promising antibacterial agents against resistant Gram-positive pathogens.
Eur J Med Chem
; 165: 133-141, 2019 Mar 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-30665143
11.
Two independent ways of preparing hypercharged hydrolyzable polyaminorotaxane.
Biomacromolecules
; 9(7): 2007-13, 2008 Jul.
Artigo
em Inglês
| MEDLINE | ID: mdl-18517251
12.
Synthesis of 3-phenylnaphthalenic derivatives as new selective MT(2) melatoninergic ligands.
Bioorg Med Chem
; 16(18): 8339-48, 2008 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-18778943
13.
Design and synthesis of benzofuranic derivatives as new ligands at the melatonin-binding site MT3.
Bioorg Med Chem
; 16(9): 4954-62, 2008 May 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-18372181
14.
Design, synthesis and biological evaluation of novel ring-opened cromakalim analogues with relaxant effects on vascular and respiratory smooth muscles and as stimulators of elastin synthesis.
Eur J Med Chem
; 144: 774-796, 2018 Jan 20.
Artigo
em Inglês
| MEDLINE | ID: mdl-29291445
15.
Traditional uses, phytochemistry and pharmacological properties of African Nauclea species: A review.
J Ethnopharmacol
; 212: 106-136, 2018 Feb 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-29045823
16.
Make azoles active again: chalcones as potent reversal agents of transporters-mediated resistance in Candida albicans.
Future Med Chem
; 10(18): 2177-2186, 2018 Sep 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-30043631
17.
Piperidinyl-embeded chalcones possessing anti PI3Kδ inhibitory properties exhibit anti-atopic properties in preclinical models.
Eur J Med Chem
; 158: 405-413, 2018 Oct 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-30237123
18.
Ferrocene-embedded flavonoids targeting the Achilles heel of multidrug-resistant cancer cells through collateral sensitivity.
Eur J Med Chem
; 130: 346-353, 2017 Apr 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-28273561
19.
New, highly potent and non-toxic, chromone inhibitors of the human breast cancer resistance protein ABCG2.
Eur J Med Chem
; 122: 291-301, 2016 Oct 21.
Artigo
em Inglês
| MEDLINE | ID: mdl-27376492
20.
Synthesis and pharmacological evaluation of dual ligands for melatonin (MT1/MT2) and serotonin 5-HT2C receptor subtypes (II).
Eur J Med Chem
; 90: 822-33, 2015 Jan 27.
Artigo
em Inglês
| MEDLINE | ID: mdl-25528336