Detalhe da pesquisa
1.
Promising aryl selenoate derivatives as antileishmanial agents and their effects on gene expression.
Antimicrob Agents Chemother
; 68(4): e0155923, 2024 Apr 03.
Artigo
em Inglês
| MEDLINE | ID: mdl-38497616
2.
Novel Pitolisant-Derived Sulfonyl Compounds for Alzheimer Disease.
Int J Mol Sci
; 25(2)2024 Jan 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-38255872
3.
Examination of multiple Trypanosoma cruzi targets in a new drug discovery approach for Chagas disease.
Bioorg Med Chem
; 58: 116577, 2022 03 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-35189560
4.
Rational modification of Mannich base-type derivatives as novel antichagasic compounds: Synthesis, in vitro and in vivo evaluation.
Bioorg Med Chem
; 27(17): 3902-3917, 2019 09 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-31345745
5.
Library of Seleno-Compounds as Novel Agents against Leishmania Species.
Antimicrob Agents Chemother
; 61(6)2017 06.
Artigo
em Inglês
| MEDLINE | ID: mdl-28320721
6.
In vitro antileishmanial activity and iron superoxide dismutase inhibition of arylamine Mannich base derivatives.
Parasitology
; 144(13): 1783-1790, 2017 Nov.
Artigo
em Inglês
| MEDLINE | ID: mdl-28789716
7.
Design and synthesis of novel quinoxaline derivatives as potential candidates for treatment of multidrug-resistant and latent tuberculosis.
Bioorg Med Chem Lett
; 26(9): 2188-93, 2016 May 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-27025343
8.
Synthesis and biological evaluation of quinoxaline di-N-oxide derivatives with in vitro trypanocidal activity.
Bioorg Med Chem Lett
; 26(3): 903-906, 2016 Feb 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-26750255
9.
Synthesis, biological evaluation and structure-activity relationships of new quinoxaline derivatives as anti-Plasmodium falciparum agents.
Molecules
; 19(2): 2166-80, 2014 Feb 18.
Artigo
em Inglês
| MEDLINE | ID: mdl-24552985
10.
New amide derivatives of quinoxaline 1,4-di-N-oxide with leishmanicidal and antiplasmodial activities.
Molecules
; 18(4): 4718-27, 2013 Apr 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-23609622
11.
Neglected Zoonotic Diseases: Advances in the Development of Cell-Penetrating and Antimicrobial Peptides against Leishmaniosis and Chagas Disease.
Pathogens
; 12(7)2023 Jul 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-37513786
12.
New quinoxaline derivatives as potential MT1 and MT2 receptor ligands.
Molecules
; 17(7): 7737-57, 2012 Jun 25.
Artigo
em Inglês
| MEDLINE | ID: mdl-22732886
13.
Antiplasmodial and leishmanicidal activities of 2-cyano-3-(4-phenylpiperazine-1-carboxamido) quinoxaline 1,4-dioxide derivatives.
Molecules
; 17(8): 9451-61, 2012 Aug 07.
Artigo
em Inglês
| MEDLINE | ID: mdl-22871647
14.
Potential of sulfur-selenium isosteric replacement as a strategy for the development of new anti-chagasic drugs.
Acta Trop
; 233: 106547, 2022 Sep.
Artigo
em Inglês
| MEDLINE | ID: mdl-35667455
15.
New 1,4-di-N-oxide-quinoxaline-2-ylmethylene isonicotinic acid hydrazide derivatives as anti-Mycobacterium tuberculosis agents.
Bioorg Med Chem Lett
; 21(12): 3699-703, 2011 Jun 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-21570839
16.
New salicylamide and sulfonamide derivatives of quinoxaline 1,4-di-N-oxide with antileishmanial and antimalarial activities.
Bioorg Med Chem Lett
; 21(15): 4498-502, 2011 Aug 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-21724395
17.
Aryl piperazine and pyrrolidine as antimalarial agents. Synthesis and investigation of structure-activity relationships.
Exp Parasitol
; 128(2): 97-103, 2011 Jun.
Artigo
em Inglês
| MEDLINE | ID: mdl-21354139
18.
Trypanocidal properties, structure-activity relationship and computational studies of quinoxaline 1,4-di-N-oxide derivatives.
Exp Parasitol
; 127(4): 745-51, 2011 Apr.
Artigo
em Inglês
| MEDLINE | ID: mdl-21272583
19.
Studies on log Po/w of quinoxaline di-N-oxides: a comparison of RP-HPLC experimental and predictive approaches.
Molecules
; 16(9): 7893-908, 2011 Sep 13.
Artigo
em Inglês
| MEDLINE | ID: mdl-22143549
20.
Design and synthesis of Mannich base-type derivatives containing imidazole and benzimidazole as lead compounds for drug discovery in Chagas Disease.
Eur J Med Chem
; 223: 113646, 2021 Nov 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-34182359